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AL-438 is a potent, selective and orally active glucocorticoid receptor modulator with Kis of 2.5, 1786, 53, 1440, >1000 nM for glucocorticoid receptor, progesterone receptor, mineralocorticoid receptor, androgen receptor, estrogen receptor, respectively. AL-438 shows antiinflammatory activity.
| Molecular Weight | 347.45 |
| Formula | C23H25NO2 |
| CAS Number | 239066-73-0 |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
[4] Jonathan Rosen, et al. Endocr Rev. The search for safer glucocorticoid receptor ligands
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