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Phospholipase Phospholipase (e.g. PLA)

Inhibitors

Cat.No.  Name Information
M6074 AA26-9 AA26-9 is a potent and broad spectrum serine hydrolase inhibitor.
M21360 (E/Z)-Polydatin (E/Z)-Polydatin (E/Z)-Piceid) is a single-crystal compound originally isolated from the roots and rhizomes of Echinacea purpurea with antiplatelet aggregation, anti-low density lipoprotein (LDL) oxidation, cardioprotective, anti-inflammatory and immunomodulatory properties.
M20582 ST 271 ST271 is a tyrphostin-like protein tyrosine kinase (PTK) inhibitor which inhibits phospholipase D (PLD) activity.
M14515 Varespladib methyl Varespladib methyl (A-002; LY333013) is a selective inhibitor of group II secretory phospholipase A2 (PLA2).
M14514 N-(p-amylcinnamoyl) Anthranilic Acid N-(p-amylcinnamoyl) Anthranilic Acid (ACA) is a broad spectrum Phospholipase A2 (PLA2) inhibitor and TRP channel blocker.
M14513 Melittin TFA Melittin TFA is a PLA2 activator, stimulates the activity of the low molecular weight PLA2, while it does not the increase activity of the high molecular weight PLA2.
M14512 MAFP MAFP (Methyl Arachidonyl Fluorophosphonate) is an selective, active-site directed and irreversible inhibitor of cPLA2 and iPLA2. MAFP is also a potent irreversible inhibitor of anandamide amidase.
M14511 LEI-401 LEI-401 is a first-in-class, selective, and CNS-active NAPE-PLD (N-acylphosphatidylethanolamine phospholipase D) inhibitor, with an IC50 of 27 nM. LEI-401 modulates emotional behavior in mice.
M14510 D609 D609 is a selective competitive inhibitor of phosphatidyl choline-specific phospholipase C (PC-PLC), with Ki of 6.4 μM.
M14509 CAY10650 CAY10650 is a highly potent cytosolic phospholipase A2α (cPLA2α) inhibitor with an IC50 value of 12 nM. CAY10650 suppresses lipid droplets formation and PGE2 secretion.
M14508 3-Nitrocoumarin 3-Nitrocoumarin (3-NC) is a potent and selective Phospholipase C-γ (PLC-γ) inhibitor.
M8927 VU-0155069 VU-0155069 is a potent and selective phospholipase D1 (PLD1) inhibitor.
M6074 AA26-9 AA26-9 is a potent and broad spectrum serine hydrolase inhibitor.
M5201 FIPI FIPI inhibited both PLD1 and PLD2 in a dose-dependent manner, with 50% loss of activity observed at approximately 25 nM.
M5170 U73122 U73122 is a potent inhibitor of phospholipase C, phospholipase A2 and 5-LO (5-lipoxygenase).
M4144 Tanshinone-I Tanshinone-I
M3969 Polydatin Polydatin is a monocrystaline compound isolated from Polygonum cuspidatum Sieb. et Zucc. (Polygonaceae) with biological properties, such as anti-inflammation, anti-oxidative and nephroprotective effects.
M2759 Darapladib Darapladib is a selective and orally active inhibitor of Lp-PLA2 with IC50 of 270 pM.
M1935 LY315920 LY315920 is a potent, selective inhibitor of recombinant human, group IIA, nonpancreatic secretory PLA2 (sPLA2).



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