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PAR Protease-Activated Receptor

Cat.No.  Name Information
M8538 ML354 ML354 is a potent and selective PAR4 (protease activated receptor-4) antagonist.
M49480 NRD-21 NRD-21 is an allosteric inhibitor of PAR1 Gq signaling, with IC50 of 0.38 uM in intracellular calcium mobilization assay. NRD-21 has improved anti-Inflammatory activity and is much more plasma stable than ML161, it is a promising lead compound for the parmodulin class for anti-thrombotic and anti-inflammatory indications research.
M31169 Parstatin (mouse) TFA Parstatin (mouse) TFA is a peptide formed by protein hydrolysis upon PAR1 receptor activation and is also a PAR-1 agonist with cellular permeability. In addition, Parstatin (mouse) TFA is also a potent inhibitor of angiogenesis. It can be used in studies related to ischemia-reperfusion injury.
M31168 TFLLR-NH2 (TFA) TFLLR-NH2 (TFA) is a selective protease-activated receptor 1 (PAR1) agonist with an EC50 value of 1.9 μM.
M21516 PZ-128 PZ-128 (P1pal-7), a cell-penetrating peptide, is a first-in-class, specific and reversible protease activating receptor 1 (PAR1) antagonist. It has anti-platelet, anti-metastasis, anti-angiogenesis and anticancer effects.
M14047 FSLLRY-NH2 TFA FSLLRY-NH2 TFA is a protease-activated receptor 2 (PAR2) inhibitor.
M10238 PAR-2 (6-1) amide (human) VKGILS-NH2 is a reversed amino acid sequence control peptide for SLIGKV-NH2.
M10237 Protease-Activated Receptor-2, amide Protease-Activated Receptor-2, amide (SLIGKV-NH2) is a highly potent agonist of PAR2 with IC50 of 10.4 uM.
M10236 PAR-2 (1-6) (mouse, rat) PAR-2 (1-6) (mouse, rat) is a PAR2 activator, it can be used to explore signaling through PAR2 in cells.
M10235 SLIGRL-NH2 SLIGRL-NH2 (Protease-Activated Receptor-2 Activating Peptide) is an agonist of Protease-Activated Receptor-2 (PAR-2).
M10143 AZ3451 AZ3451 is a potent PAR2 (protease-activated receptor-2) antagonist with IC50 of 23 nM, which plays a part in inflammation response, apoptosis, autophagy and cellular senescence during Osteoarthritis (OA).
M9814 (Ala1)-PAR-4 (1-6) (mouse) (Ala1)-PAR-4 (1-6) (mouse)
M9813 PAR-4 (1-6) (mouse) PAR-4 (1-6) (mouse)
M9812 PAR-4 (1-6) (human) PAR-4 (1-6) (human) is an N-terminal fragment of protease-activated receptor 4 (PAR4) that acts as a PAR4 agonist.
M6243 Vorapaxar Sulfate Vorapaxar is a first-in-class, potent and orally-active protease-activated receptor 1 (PAR-1) antagonist that blocks thrombin-mediated platelet activation without interfering with thrombin-mediated fibrin deposition.
M3123 Vorapaxar Vorapaxar (SCH 530348) is a potent and orally active thrombin receptor (PAR-1) antagonist with Ki of 8.1 nM.
M2574 ML161 Parmodulin 2 (ML161) is an allosteric inhibitor of PAR1 with IC50 of 0.26 μM.
M54466 TRAP-6 amide TRAP-6 amide is a PAR-1 thrombin receptor agonist peptide.
M54429 Protease-Activated Receptor-1, PAR-1 Agonist Protease-Activated Receptor-1, PAR-1 Agonist is a selective proteinase-activated receptor1 (PAR-1) agonist peptide.
M54388 FSLLRY-NH2 FSLLRY-NH2 is a protease-activated receptor 2 (PAR2) inhibitor.




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