PAR Protease-Activated Receptor

Cat.No.	Name	Information
M8538	ML354	ML354 is a potent and selective PAR4 (protease activated receptor-4) antagonist.
M21101	BMS-986120	BMS-986120 is a first-in-class oral protease-activated receptor 4 (PAR4) inhibitor with IC50 values of 9.5 nM in human and 2.1 nM in monkey blood.BMS-986120 exhibits potent and selective antiplatelet effects. BMS-986120 has potent and selective antiplatelet effects and can be used in studies related to arterial thrombosis.
M14050	SCH79797	SCH79797 is a highly potent, selective nonpeptide protease activated receptor 1 (PAR1) antagonist.
M14049	PAR-4 Agonist Peptide, amide TFA	PAR-4 Agonist Peptide, amide TFA (PAR-4-AP TFA; AY-NH2 TFA) is a proteinase-activated receptor-4 (PAR-4) agonist, which has no effect on either PAR-1 or PAR-2 and whose effects are blocked by a PAR-4 antagonist.
M14048	GB-88	GB-88 is an oral, selective non-peptide antagonist of PAR2, inhibits PAR2 activated Ca²⁺ release with an IC50 of 2 µM.
M10777	AGN 194310	AGN 194310 (VTP-194310) is a highly affinity, potent, selective pan antagonist of retinoic acid receptors (RARs) against RARα, RARβ, RARγ Kd The values are 3 nM, 2 nM, and 5 nM, respectively.