| Cat.No. | Name | Information |
|---|---|---|
| M2206 | TH-302 (Evofosfamide) | TH-302 is a highly potent and selective hypoxia-activated procompound targeting hypoxic regions of solid tumors with IC50 of 19 nM. |
| M6098 | Baicalein | Baicalein is a CYP2C9 and prolyl endopeptidase inhibitor, IC50 value of 3.12 mM. |
| M9325 | EGTA | EGTA is a specific calcium chelator with a Kd of 60.5 nM at physiological pH (7.4) and a high specificity for Ca2+ than for Mg2+.EGTA significantly inhibits the substrate adhesion capacity of inflammatory macrophages. |
| M9330 | Brij-35 | Brij-35 (Polidocanol) is a high HLB, ethoxylated, nonionic ether of lauryl alcohol with broad pH stability. |
| M6154 | 2-PMPA tetrasodium | 2-PMPA (PMPA tetrasodium salt) is a potent and selective inhibitor of glutamate carboxypeptidase II (GCPII) with an IC50 of 300 pM. |
| M2250 | Pamidronate disodium | Pamidronate disodium is a nitrogen containing bisphosphonate, used to prevent osteoporosis. |
| M9916 | DPPH | DPPH (2,2-Diphenyl-1-picrylhydrazyl) is a stable free radical that measures the free radical scavenging activity of antioxidants. |
| M9194 | Insulin (human) | Insulin (human) is a polypeptide hormone that regulates the level of sugar (glucose) in the blood and is produced by beta cells of islets. |
| M3409 | Formestane | Formestane is a second generation selective aromatase inhibitor with an IC50 of 80 nM. |
| M9331 | 10-Hydroxy-trans-2-decenoic acid | 10-hydroxy-2-decenoic acid (10-H2DA) is the principal lipid component in royal jelly which is the food for queen and larvae honeybees. |
| M11043 | DJ001 | DJ001 is a highly specific, selective and non-competitive protein tyrosine phosphatase-σ (PTPσ) inhibitor,IC50 is 1.43 μM. DJ001 has no inhibitory activity against other phosphatases and only moderate inhibitory activity against protein phosphatase 5. DJ001 Promotes hematopoietic stem cell regeneration. |
| M11042 | ASK1-IN-2 | ASK1-IN-2 is a potent, orally active apoptosis signal-modulating kinase 1 (ASK1) inhibitor,IC50 The value is 32.8 nM. |
| M11036 | L-Ascorbic acid 2-phosphate | L-ascorbic acid 2-phosphate is a long-acting vitamin C derivative that stimulates collagen expression and formation. L-ascorbic acid 2-phosphate increases alkaline phosphatase (ALP) activity and runx2A expression in hASC during osteoblast differentiation. |
| M11035 | L-Perillaldehyde | |
| M11004 | GSK-2324 | GSK2324 is a FXR agonist with EC50 value of 50 nM. |
| M11003 | Benpyrine | Benpyrine is a highly specific orally active TNF-α inhibitor.KD The value is 82.1 μM. Benpyrine binds tightly to TNF-α and blocks its interaction with TNFR1,IC50 The value is 0.109 μM. |
| M10963 | ARCC-4 | ARCC-4 is based on PROTAC technology, a nanomolar grade androgen receptor (AR) degrader D50 The value is 5 nM. ARCC-4 is an AR PROTAC recruited by von Hippel-Lindau (VHL) based on enzalutamide. ARCC-4 effectively degrades AR mutations associated with antiandrogen studies. |
| M10962 | RU 59063 | RU 59063 is a prototype of high-affinity nonsteroidal androgen receptor (AR) ligands. |
| M10950 | SPD304 | SPD304 is a selective inhibitor of tumor necrosis factor α (TNF-α) that promotes the separation of tumor necrosis factor trimers, thereby blocking their interaction with receptors. SPD304 inhibits tumor necrosis factor in vitro α and receptor 1 binding IC50 The value is 22 μM. |
| M10949 | C 87 | C87 is a novel small molecule inhibitor of TNFα; Efficient inhibition of TNFα-induced cytotoxicity,IC50 The value is 8.73 μM. |
| M10947 | INT-767 | INT-767 is a farnidol X receptor (FXR)/TGR5 dual agonist,EC50 The values are 30 and 630 nM, respectively. |
| M10946 | Glyco-Obeticholic acid | Glyco-obeticholic acid is an active metabolite of taurine. Obeticholic Acid is an oral bioavailable fancy-like X receptor (FXR) agonist. |
| M10944 | BT-13 | BT-13 is a potent, glial-derived neurotrophic factor (GDNF) receptor RET selective agonist (independent of GDNF ligands) that promotes the growth of process ninsters in vitro sensory neurons and mitigates the occurrence of neuropathy in rats. |
| M10912 | asukamycin | |
| M10911 | ZXH-3-26 | ZXH-3-26 is a PROTAC connected by the Cereblon ligand and brd4 ligands, and after 5 hours of processing,DC50 Approximately 5 nM. |
| M10904 | Angstrom6 | Angstrom6 (A6 Peptide) is an 8-amino acid peptide derived from single-stranded urokinase plasminogen activator (scuPA) that interferes with the uPA/uPAR cascade and eliminates downstream effects. Angstrom6 binds to CD44 to inhibit migration, invasion and metastasis of tumor cells and regulate CD44-mediated cell signaling. |
| M10901 | viloxazine | |
| M10895 | Umirolimus | Umirolimus, a derivative of macrotriene lactone Rapamycin, is a powerful immunosuppressant and anti-inflammatory agent. Umirolimus is highly lipophilic and can be used as a drug-eluting stent. |
| M10893 | Tesetaxel | |
| M10891 | Taranabant | Taranabant is a potent and selective cannabinoid 1 (CB1) receptor reverse agonist that inhibits binding and the functional activity of multiple agonists, acting on human CB1R,Ki 0.13 nM. |
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