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Abmole Inhibitor Catalog 2017

Estrogen Receptor Estrogen Receptor

Inhibitors

Cat.No.  Name Information
M5599 Drospirenone Drospirenone is a synthetic progestin that is an analog to spironolactone.
M5564 Desogestrel Desogestrel is a synthetic progestational hormone used often as the progestogenic component of combined oral contraceptive agents.
M5511 Chlormadinone acetate Chlormadinone acetate is a steroidal progestin with additional antiandrogen and antigonadotropic effects, used often in combinations as an oral contraceptive. Its half-life is about 34-38 hours.
M4836 G-1 G-1 is a potent and selective GPR30 receptor agonist (Ki = 11 nM, EC50 = 2 nM).
M4835 DPN DPN is a highly potent estrogen ERβ receptor agonist with a 70-fold selectivity over ERα with EC50 values are 0.85 and 66 nM,respectively.
M4834 PPT PPT is a potent subtype-selective estrogen receptor agonist with EC50 ~ 200 pM and displays 410-fold selectivity for ERα over ERβ.
M3945 Estrone Estrone is an estrogenic hormone.
M3764 DY131 DY131(GSK 9089) is a novel selective agonist of ERRβ and ERRγ which displays minimal activity at ERRα, ERα and ERβ at concentrations up to 30 μM.
M3652 Ospemifene Ospemifene is a non-hormonal selective estrogen receptor modulator (SERM) which is used for the treatment of dyspareunia.
M3564 Clomifene citrate Clomifene citrate is a selective estrogen receptor modulator.
M3392 Ethinyl Estradiol Ethinyl Estradiol is an orally bio-active estrogen used in almost all modern formulations of combined oral contraceptive pills.
M3371 Estriol Estriol is an antagonist of the G-protein coupled estrogen receptor in estrogen receptor-negative breast cancer cells.
M2097 LY500307 LY500307 is a potent, selective estrogen receptor beta agonist with an EC50 of 0.66 nM.
M1966 Fulvestrant Fulvestrant (Faslodex) is a novel estrogen receptor (ER) antagonist (IC50 = 0.29 nM).


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