| Cat.No. | Name | Information |
|---|---|---|
| M1966 | Fulvestrant | Fulvestrant is a Estrogen receptor (ER) antagonist with IC50 of 0.094 nM. Fulvestrant can also induce autophagy and apoptosis, and has anti-tumor effect. |
| M3371 | Estriol | Estriol is an antagonist of the G-protein coupled estrogen receptor in estrogen receptor-negative breast cancer cells. |
| M4368 | Kaempferol | Kaempferol is an inverse agonist of ERRα and ERRγ that inhibits estrogen receptor (ER α) expression in breast cancer cells and induces apoptosis by activating MEK-MAPK in glioblastoma cells and lung cancer cells. It can be used in breast cancer research. |
| M7353 | Tamoxifen | Tamoxifen is an orally active, selective estrogen receptor partial agonist/antagonist. Tamoxifen is a potent Hsp90 activator and enhances the Hsp90 molecular chaperone ATPase activity. Tamoxifen also potent inhibits infectious EBOV Zaire and Marburg (MARV) with IC50 of 0.1 µM and 1.8 µM, respectively. |
| M7871 | G15 | G15 is a high affinity and selective G-protein-coupled estrogen receptor (GPER/GPR30) antagonist with a Ki of 20 nM. |
| M4374 | Gypenoside-XVII | Gypenoside XVII is a novel phytoestrogens belonging to gypenosides, which can activate estrogen receptors. |
| M2174 | Calcitriol | Calcitriol is an Active metabolite of vitamin D3 that activates the vitamin D receptor. *The compound is unstable in solutions, freshly prepared is recommended |
| M4836 | G-1 | G-1 is a potent and selective GPR30 receptor agonist (Ki = 11 nM, EC50 = 2 nM). |
| M8508 | PHTPP | PHTPP is a selective estrogen receptor β (ERβ) full antagonist with 36-fold selectivity for ERβ over ERα. |
| M10348 | 27-Hydroxycholesterol | 27-Hydroxycholesterol is a selective estrogen receptor modulator, and it is also an agonist of the liver X receptor. |
| M50377 | Yp537 | Yp537 is an estrogen receptor (ER) inhibitor that blocks dimerization of the human estrogen receptor. |
| M45361 | Palazestrant | Palazestrant is a novel, orally active, estrogen receptor antagonist and selective estrogen receptor degrader. It can be used in studies related to ER+/HER2+ breast cancer. |
| M45336 | Acolbifene hydrochloride | Acolbifene hydrochloride is an active metabolite of EM800 and an orally available, selective estrogen receptor modulator (SERM) that inhibits estradiol-induced ERα (IC50 = 2 nM) and ERβ (IC50 = 0.4 nM) transcriptional activity, has significant anti-estrogenic effects on the mammary gland and uterus, and has anticancer activity. possesses anticancer activity. |
| M45335 | Acolbifene | Acolbifene is an active metabolite of EM800 and an orally active pure anti-estrogen and selective estrogen receptor (ER) antagonist that inhibits estradiol-induced ERα (IC50 = 2 nM) and ERβ (IC50 = 0.4 nM) transcriptional activity and has anticancer activity. |
| M45334 | Zearalanone | Zearalanone is a nonsteroidal estrogenic mycotoxin produced by a Fusarium genus, Fusarium, that grows in several cereal grains and has low acute toxicity and carcinogenicity.Zearalenone is agonistic to the estrogen receptor (ER), exhibits marked estrogenic and anabolic properties in several animals, and can have serious effects on the reproductive system of animals. . |
| M44724 | 3'-Hydroxymirificin | 3'-Hydroxymirificin is a naural compound that can be isolated from Pueraria lobata roots. |
| M43603 | ERα degrader 6 | ERα degrader 6 is an ERα degrader (KI: 75 nM). |
| M43602 | ER degrader 5 | ER degrader 5 is a potent estrogen receptor (ER) degrader. |
| M43601 | ER degrader 6 | ER degrader 6 is a potent Estrogen Receptor (ER)α degrader. |
| M43600 | Estrogen receptor modulator 7 | Estrogen receptor modulator 7 is a potent estrogen receptor modulator. |
| M43599 | ER degrader 4 | ER degrader 4 is a selective and orally active estrogen receptor degrader. |
| M43598 | SLU-PP-1072 | SLU-PP-1072 is a dual ERRα/γ inverse agonist, used in Prostate cancer (PCa) research. |
| M43597 | ERRγ agonist-2 | ERRγ agonist-2 is a potent and selective ERRγ inverse agonist with a Kd value of 6.5 μM. |
| M43596 | Yp537 TFA | Yp537 TFA is an estrogen receptor (ER) inhibitor that blocks dimerization of the human estrogen receptor. |
| M43595 | Estrogen receptor modulator 8 | Estrogen receptor modulator 8 is an orally active inhibitor of Estrogen Receptor/ERR α (IC50=0.437 nM, MCF-7 cells). |
| M43594 | Estrogen receptor antagonist 8 | Estrogen receptor antagonist 8 is a potent estrogen receptor ER antagonist with an EC50 of 4.160 μM. |
| M43593 | SLU-PP-332 | SLU-PP-332 is a pan-Estrogen Receptor/ERR agonist with EC50 values of 98, 230 and 430 nM for ERRα, ERRβ and ERRγ, respectively. |
| M43592 | ET receptor antagonist 3 | ET receptor antagonist 3 is an orally active ET receptor antagonist (IC50=0.26 nM), which can be used for research in pulmonary arterial hypertension (PAH). |
| M43591 | ET receptor antagonist 2 | ET receptor antagonist 2 is an orally active ET receptor antagonist (IC50=0.22 nM), which can be used for research in pulmonary arterial hypertension (PAH). |
| M43590 | ET receptor antagonist 1 | ET receptor antagonist 1 is an orally active ET receptor antagonist (IC50=0.18 nM), which can be used for research in pulmonary arterial hypertension (PAH). |
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