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Estrogen Receptor Estrogen Receptor

Cat.No.  Name Information
M1966 Fulvestrant Fulvestrant is a Estrogen receptor (ER) antagonist with IC50 of 0.094 nM. Fulvestrant can also induce autophagy and apoptosis, and has anti-tumor effect.
M3371 Estriol Estriol is an antagonist of the G-protein coupled estrogen receptor in estrogen receptor-negative breast cancer cells.
M4368 Kaempferol Kaempferol is an inverse agonist of ERRα and ERRγ that inhibits estrogen receptor (ER α) expression in breast cancer cells and induces apoptosis by activating MEK-MAPK in glioblastoma cells and lung cancer cells. It can be used in breast cancer research.
M7353 Tamoxifen Tamoxifen is a estrogen receptor partial agonist/antagonist.
M7871 G15 G15 is a high affinity and selective G-protein-coupled estrogen receptor (GPER/GPR30) antagonist with a Ki of 20 nM.
M4374 Gypenoside-XVII Gypenoside XVII is a novel phytoestrogens belonging to gypenosides, which can activate estrogen receptors.
M2174 Calcitriol Calcitriol is an Active metabolite of vitamin D3 that activates the vitamin D receptor. *The compound is unstable in solutions, freshly prepared is recommended
M4836 G-1 G-1 is a potent and selective GPR30 receptor agonist (Ki = 11 nM, EC50 = 2 nM).
M8508 PHTPP PHTPP is a selective estrogen receptor β (ERβ) full antagonist with 36-fold selectivity for ERβ over ERα.
M10348 27-Hydroxycholesterol 27-Hydroxycholesterol is a selective estrogen receptor modulator, and it is also an agonist of the liver X receptor.
M7493 XCT 790 XCT 790 is a potent, selective ERRα inverse agonist with an IC50 value of 0.37 μM and is inactive against ERRγ and estrogen receptors ERα and ERβ.
M7483 WAY 200070 WAY 200070 is a selective ERβ agonist.
M6717 ERB 041 ERB 041 is a potent and selective estrogen receptor β (ERβ) agonist, with IC50s of 5.4, 3.1, and 3.7 nM for ERβ in humans, rats, and mice, respectively.ERB 041 is more than 200 times more selective for ERβ than for ERα. In addition, ERB 041 inhibits the WNT/β-catenin signaling pathway and induces apoptosis in ovarian cancer cells.
M6710 Endoxifen Z-isomer hydrochloride Endoxifen Z-isomer hydrochloride is a Tamoxifen metabolite and a potent estrogen receptor (ER) antagonist that concentration-dependently inhibits hERG with an IC50 value of 1.6 μM.
M6165 GSK 4716 GSK 4716 is a selective agonist with estrogen-related receptors ERRβ and ERRγ.
M6083 AZD9496 AZD9496 is an oral estrogen receptor inhibitor that blocks the growth of ER-positive and ESR1 mutant breast tumours in preclinical models.
M6069 β-Estradiol 17-acetate β-Estradiol 17-acetate is a metabolite of estradiol.
M5917 Raloxifene HCl RaloxifeneHcl(LY156758 Hcl) is a second generation selective estrogen receptor antagonist.
M5765 Megestrol Acetate Megestrol acetate is a synthetic progestogen, used to treat breast cancer and loss of appetite.
M5698 Hydroxyprogesterone caproate Hydroxyprogesterone Caproate is a synthetic progesterone receptor (PR) agonist that binds and activates the nuclear progesterone receptor in the reproductive system and may be used in studies related to genitourinary disorders.
M5668 Bavachin Bavachin, a flavonoid first isolated from seeds of P. corylifolia, acts as a phytoestrogen that activates the estrogen receptors ERα and ERβ with EC50s of 320 and 680 nM, respectively.
M5635 Etonogestrel Etonogestrel is a synthetic form of the naturally occurring female sex hormone progesterone. It binds to the cytoplasmic progesterone receptors in the reproductive system and subsequently activates progesterone receptor mediated gene expression.
M5628 Ethisterone Ethisterone is a progestogen hormone being considered to treat prostate cancer.
M5627 Estropipate Estropipate is a form of estrogen, used to treat symptoms of menopause, also used to prevent osteoporosis.
M5599 Drospirenone Drospirenone is a synthetic progestin that is an analog to spironolactone.
M5564 Desogestrel Desogestrel is a synthetic progestational hormone used often as the progestogenic component of combined oral contraceptive agents.
M5511 Chlormadinone acetate Chlormadinone acetate is a steroidal progestin with additional antiandrogen and antigonadotropic effects, used often in combinations as an oral contraceptive. Its half-life is about 34-38 hours.
M5434 Avobenzone Avobenzone is an oil soluble ingredient used in sunscreen products to absorb the full spectrum of UVA rays and a dibenzoylmethane derivative.
M4835 DPN DPN is a highly potent estrogen ERβ receptor agonist with a 70-fold selectivity over ERα with EC50 values are 0.85 and 66 nM,respectively.
M4834 Propyl pyrazole triol (PPT) PPT is a potent subtype-selective estrogen receptor agonist with EC50 ~ 200 pM and displays 410-fold selectivity for ERα over ERβ.




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