About 22 results found for searched term "SP-10" (0.114 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M3358 | Procainamide hydrochloride | Sodium Channel |
| Procaine amide hydrochloride; SP 100 hydrochloride | ||
| Procainamide hydrochloride is a sodium channel blocker, and also a DNA methyltransferase inhibitor. | ||
| M5398 | Aliskiren Hemifumarate | Renin |
| CGP 60536; CGP60536B; SPP 100 | ||
| Aliskiren hemifumarate is a direct renin inhibitor with IC50 of 1.5 nM. | ||
| M8245 | SPV-106 | Others |
| SPV106 is a mixed inhibitor/activator of histone acetyltransferase (HAT) activity. | ||
| M9794 | Ebselen | Calcium Channel |
| SPI-1005; PZ-51; CCG-39161 | ||
| Ebselen (SPI-1005) is a potent voltage-dependent calcium channel (VDCC) blocker. Ebselen is an inhibitor of HIV-1 capsid CTD dimerization. Ebselen can permeate the blood-brain barrier and has anti-inflammatory, antioxidant and anticancer activity | ||
| M10565 | Kisspeptin-10, human TFA | Peptides |
| KP-10; Tyr-Asn-Trp-Asn-Ser-Phe-Gly-Leu-Arg-Phe-NH2 | ||
| Kisspeptin-10, human TFA is a potent vasoconstrictor and inhibitor of angiogenesis, it acts as a tumor metastasis suppressor via its receptor GPR54. | ||
| M10724 | Pridopidine | Dopamine Receptor |
| ACR16; ASP2314; FR310826 | ||
| Pridopidine is a dopamine (DA) stabilizer that acts as a low-affinity dopamine D2 receptor (D2R) antagonist. Pridopidine high affinity acts on sigma 1 receptor (S1R),Ki Values of 70 to 80 nM are approximately 100 times higher than their affinity for D2R. | ||
| M13693 | Taltobulin | Microtubule |
| HTI-286; SPA-110 | ||
| Taltobulin (HTI-286), a synthetic analogue of the tripeptide hemiasterlin, is a potent antimicrotubule agent that circumvents P-glycoprotein-mediated resistance in vitro and in vivo. | ||
| M13694 | Taltobulin hydrochloride | Microtubule |
| HTI-286 hydrochloride; SPA-110 hydrochloride | ||
| Taltobulin hydrochloride (HTI-286 hydrochloride), a synthetic analogue of the tripeptide hemiasterlin, is a potent antimicrotubule agent that circumvents P-glycoprotein-mediated resistance in vitro and in vivo. | ||
| M13816 | Procainamide | DNA Methyltransferase |
| Procaine amide; SP 100 | ||
| Procainamide is a specific and potent inhibitor of DNA methyltransferase 1 (DNMT1). Procainamide is a Class 1A antiarrhythmic agent. Procainamide has the potential for the research of cancer and arrhythmias. | ||
| M14530 | Aliskiren | Renin |
| CGP 60536; CGP60536B; SPP 100 | ||
| Aliskiren(CGP 60536) is a direct renin inhibitor with IC50 of 1.5 nM. | ||
| M14582 | Itanapraced | Gamma-secretase/Beta-secretase |
| CHF5074; CSP-1103 | ||
| Itanapraced (CHF5074) is a novel γ-secretase modulator, reduces Aβ42 and Aβ40 secretion, with an IC50 of 3.6 and 18.4 μM, respectively. | ||
| M28589 | SP-100030 | NF-κB |
| SP-100030 is a potent NF-κB and activator protein-1 (AP-1) double inhibitor (IC50s=50 and 50 nM, respectively). SP-100030 inhibits IL-2, IL-8, and TNF-alpha production in Jurkat and other T cell lines. SP-100030 decreases murine collagen-induced arthritis (CIA). | ||
| M29523 | SPL-410 | Others |
| SPL-410 is an orally active, highly potent and selective hydroxyethylamine based SPPL2a (Signal Peptide Peptidase Like 2a) inhibitor, with an IC50 of 9 nM. | ||
| M31333 | Kisspeptin-10, human ACETATE | Peptides |
| Kisspeptin-10, human ACETATE is the acetate form of Kisspeptin-10 and is also a potent vasoconstrictor and angiogenesis inhibitor that inhibits tumor metastasis through its receptor GPR54.Kisspeptin-10/GPR54 signaling through NFATc4-mediated BMP2 expression to induces osteoblast differentiation through NFATc4-mediated BMP2 expression. | ||
| M51371 | Thrombospondin-1 (1016-1021) (human, bovine, mouse) | Others |
| Thrombospondin-1 (1016-1021) (human, bovine, mouse), a Thrombospondin-1-derived peptide, is a truncated peptide devoid of CD47-binding activity. | ||
| M51669 | Cys-Arg-Gly-Asp-Phe-Pro-Ala-Ser-Ser-Cys (Disulfide bridge:cys1-cys10) | Others |
| Cys-Arg-Gly-Asp-Phe-Pro-Ala-Ser-Ser-Cys (Disulfide bridge:cys1-cys10), a decapeptide containing a cyclic RGD active sequence, is an Integrin αIIbβ3 antagonist that inhibits platelet and Adhesion of proMMP-13. | ||
| M51779 | Fmoc-Cys-Asp10 | Amino Acid Derivatives |
| Fmoc-Cys-Asp10 is a non-releasable oligopeptide linker, involves in the synthesis of releasable oligopeptide linker. | ||
| M52410 | SP-10 | AChR/AChE |
| SP-10 is a small peptide derived from S protein with an IC50 value of 1.88 nM for blocks the interaction between S protein and ACE2. | ||
| M53105 | Kisspeptin-10, rat | Others |
| Kisspeptin-10, rat is a potent vasoconstrictor and inhibitor of angiogenesis. | ||
| M54237 | Kisspeptin-10, human | Others |
| Kisspeptin-10, human is a potent vasoconstrictor and inhibitor of angiogenesis. | ||
| M54262 | Thrombospondin-1 (1016-1023) (human, bovine, mouse) | Apoptosis |
| Thrombospondin-1 (1016-1023) (human, bovine, mouse), is the C-terminal end of the native sequence of Thrombospondin-1 (TSP-1), is a CD47 agonist peptide. | ||
| M4881 | Actinomycin D | DNA/RNA Synthesis |
| Actinomycin Aiv; Dactinomycin; Act D; RASP-101 | ||
| Actinomycin D (Dactinomycin) is an antibiotic found in Streptomyces microsporum with antibacterial and anti-tumor effects. Actinomycin D is an inhibitor of RNA and protein synthesis. Actinomycin D can inhibit the protein synthesis of bacteria, directly bind to the guanine groups of single-stranded or double-stranded DNA in the transcriptional initiation complex, inhibit the activity of DNA-dependent RNA polymerase, and interfere with the transcription process of DNA, thereby inhibiting mRNA synthesis. Actinomycin D inhibits DNA repair with an IC50 value of 0.42 μM. | ||
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