About 30 results found for searched term "CP2" (0.011 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M1699 | CP-724714 | EGFR/HER2 |
| CP-724714 is a potent and selective orally active HER-2 tyrosine kinase inhibitor, IC50 = 3 nM. | ||
| M1829 | Torcetrapib | CETP |
| CP-529414 | ||
| Torcetrapib (CP-529414) is a prototype cholesteryl ester transfer protein (CETP) inhibitor with potential for decreasing atherosclerotic disease, increased cardiovascular events in clinical trials. | ||
| M1944 | CP-547632 | VEGFR/PDGFR |
| CP-547632 is a novel VEGFR-2 tyrosine kinase inhibitor with IC50 of 11 nM. | ||
| M2309 | CP-466722 | ATM/ATR |
| CP466722 | ||
| Cp-466722 is a reversible ATM inhibitor with IC50 value of 4.1 μM, but has no effect on PI3K, PIKK family proteins. | ||
| M2320 | 17-AAG (Tanespimycin) | HSP |
| Tanespimycin; 17AAG; NSC 330507; CP 127374 | ||
| 17-AAG (Tanespimycin) is a potent HSP90 inhibitor with IC50 of 5 nM. Tanespimycin depletes intracellular STK38/NDR1 and decreases STK38 kinase activity. Tanespimycin also downregulated stk38 gene expression. | ||
| M2426 | Azithromycin Dihydrate | Antibiotic |
| CP-62993 dihydrate | ||
| Azithromycin Dihydrate is an acid stable orally administered macrolide antimicrobial compound, structurally related to erythromycin. | ||
| M2612 | Danofloxacin Mesylate | Antibiotic |
| CP 76136-27 | ||
| Danofloxacin is a fluoroquinolone antibacterial for veterinary use, with MIC90 of 0.28 μM. | ||
| M3491 | OSI-420 | EGFR/HER2 |
| Desmethyl Erlotinib; CP-473420 | ||
| OSI-420 is the active metabolite of Erlotinib (EGFR inhibitor with IC50 of 2 nM). | ||
| M3505 | Glipizide | Potassium Channel |
| CP 28720; K 4024 | ||
| Glipizide is used to treat high blood sugar levels caused by a type of diabetes mellitus called type 2 diabetes. | ||
| M3526 | CPI-203 | Epigenetic Reader Domain |
| CPI203 | ||
| CPI-203 is a novel potent, selective BET bromodomain inhibitor with IC50 of 37 nM for BRD4. | ||
| M3695 | Tulathromycin A | Antibiotic |
| Tulathromycin; CP 472295 | ||
| Tulathromycin A inhibits protein synthesis by targeting bacterial ribosomes (IC50=0.26 µM). It has immunomodulatory effect. | ||
| M3872 | N-1-naphthylphthalamic acid | Plant growth regulators |
| Naphthalam; NPA; Alanape; ACP 322 | ||
| N-1-Naphthylthalamic acid is a polar auxin transport inhibitor. N-1-Naphthylthalamic acid destroys leaf initiation, KNOX protein regulation and leaf margin formation in maize. N-1-naphthylphthalic acid (NPA) is an inhibitor of IAA polar transport, it blocks auxin transport by competing with IAA for binding sites on AtPIN3. | ||
| M5261 | CP21R7 | Wnt/beta-catenin |
| CP21 | ||
| CP21R7, also known CP21, is a potent and selective GSK-3β inhibitor that can potently activate canonical Wnt signalling. | ||
| M5438 | Azithromycin | Antibiotic |
| CP 62993 | ||
| Azithromycin is an antibiotic by inhibiting protein synthesis, used for the treatment of bacterial infections. | ||
| M6259 | CP2 | Histone demethylase |
| CP2 is a cyclic peptide that inhibits the JmjC histone demethylases KDM4 with IC50 values of 42 nM and 29 nM for KDM4A and KDM4C, respectively. | ||
| M6268 | Varenicline | AChR/AChE |
| CP 526555 | ||
| Varenicline (CP 526555) is a selective α4β2 nicotinic receptor partial agonist, it stimulates nicotine receptors more weakly than nicotine itself does. | ||
| M6273 | Varenicline tartrate | AChR/AChE |
| CP 526555-18 | ||
| Varenicline Tartrate is a nicotinic AChR partial agonist, used to treat nicotine addiction. | ||
| M6629 | CP 93129 dihydrochloride | Others |
| CP 93129 dihydrochloride is a 5-HT 1B agonist. | ||
| M7340 | Sulopenem | Antibiotic |
| CP-70429 | ||
| Sulopenem is a penem antibiotic. | ||
| M7734 | CP-24879 hydrochloride | Ferroptosis |
| CP-24879 hcl | ||
| CP-24879 hydrochloride is a potent, selective and combined delta5D/delta6D desaturase inhibitor. CP-24879 (hydrochloride) can significantly reduce intracellular lipid accumulation and inflammatory injury in hepatocytes. | ||
| M7738 | CPTH2 | Histone Acetyltransferase |
| CPTH2 is a histone acetyltransferase (HAT) inhibitor modulating the Gcn5 network. | ||
| M8038 | CP-154526 hydrochloride | CRFR |
| CP-154526 hydrochloride is a selective, non-peptide antagonist of corticotropin releasing factor receptors (CRF1) with a Ki of 2.7 nM. CP 154526 hydrochloride shows selective for CRF1 over CRF2 (Ki = >10 μM). | ||
| M8039 | CP-226269 | Others |
| CP-226269 is a D4 dopamine receptor agonist with EC50 of 32 nM. | ||
| M8049 | Avridine | Adjuvants |
| CP-20961 | ||
| Avridine is a potent synthetic adjuvant that can induce arthritis in most rat strains; immunomodulator and interferon-inducing. | ||
| M8067 | CP 532623 | Others |
| CP-532623 is a potent inhbitor of cholesteryl ester transfer protein (CETP) that leads to elevated high-density lipoprotein cholesterol levels. | ||
| M8068 | CP 524515 | Others |
| CP-524515 is a potent inhbitor of cholesteryl ester transfer protein (CETP) that leads to elevated high-density lipoprotein cholesterol levels. | ||
| M8093 | Capromorelin tartrate | Ghrelin Receptor/GHSR |
| CP 424391-18 | ||
| Capromorelin tartrate is a potent ghrelin receptor agonist/growth hormone secretagogue (Ki = 7 nM). | ||
| M8103 | CP724714 | Others |
| CP724714 is a potent and selective inhibitor of HER2/ErbB2 with an IC50 value of 10 nM. | ||
| M8110 | CP-424174 | Leukotriene Receptor |
| CP-424,174 | ||
| CP-424174 is a cytokine release inhibitory compound (CRID) and also a reversible IL-1β inhibitor with an IC50 of 210 nM, which inhibits post-translational processing and secretion of IL-1β in human monocytes in the presence of LPS and ATP. | ||
| M8408 | CU-CPT22 | TLR |
| CU-CPT22 is the first probe for the complex between toll-like receptors TLR1 and TLR2. CU-CPT22 shows dose-dependent inhibitory effects blocking Pam3CSK4-induced TLR1/2 activation with an IC50 of 0.58 ± 0.09 µM. | ||
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