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VPC 23019

Cat. No. M7465

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VPC 23019 Structure

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Quality Control & Documentation
Biological Activity

VPC 23019 is a sphingosine-1-phosphate receptor antagonist. VPC 23019 inhibits S1P1 and S1P3 receptors (pKi values are 7.86 and 5.93 respectively).

Chemical Information
Molecular Weight 372.4
Formula C17H29N2O5P
CAS Number 449173-19-7
Solubility (25°C) 2eq. NaOH 18.62 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Regoli, et al. Eur J Pharmacol. Bradykinin receptors and their antagonists.

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Keywords: VPC 23019 supplier, S1P Receptor, inhibitors, activators

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