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Nelonemdaz

Cat. No. M30410

All AbMole products are for research use only, cannot be used for human consumption.

Nelonemdaz Structure
Synonym:

Salfaprodil free base; Neu2000

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Quality Control & Documentation
Biological Activity

Nelonemdaz (Salfaprodil free base) is an NR2B-selective and uncompetitive antagonist of N-methyl-D-aspartate (NMDA). Nelonemdaz is also a free radical scavenger. Nelonemdaz has excellent neuroprotection against NMDA- and free radical-induced cell death.

Chemical Information
Molecular Weight 383.22
Formula C15H8F7NO3
CAS Number 640290-67-1
Form Solid
Solubility (25°C) DMSO ≥ 112.5 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Jin Soo Lee, et al. J Stroke. The Rescue on Reperfusion Damage in Cerebral Infarction by Nelonemdaz (RODIN) Trial: Protocol for a Double-Blinded Clinical Trial of Nelonemdaz in Patients with Hyperacute Ischemic Stroke and Endovascular Thrombectomy

[2] Ji Man Hong, et al. Stroke. Nelonemdaz for Patients With Acute Ischemic Stroke Undergoing Endovascular Reperfusion Therapy: A Randomized Phase II Trial

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  Catalog
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Keywords: Nelonemdaz, Salfaprodil free base; Neu2000 supplier, GluR, inhibitors, activators

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