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Icapamespib

Cat. No. M27592

All AbMole products are for research use only, cannot be used for human consumption.

Icapamespib Structure
Synonym:

PU-HZ151

Price and Availability

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Quality Control & Documentation
Biological Activity

Icapamespib (PU-HZ151) is a potent HSP90 inhibitor with an EC50 of 5 nM. Icapamespib is able to cross blood-brain barrier.

Chemical Information
Molecular Weight 526.39
Formula C19H23IN6O2S
CAS Number 1000999-96-1
Form Solid
Solubility (25°C) DMSO ≥ 100 mg/mL
Storage Powder -20°C
References

[1] M H Silverman, et al. J Prev Alzheimers Dis. Safety, Tolerability and Pharmacokinetics of Icapamespib, a Selective Epichaperome Inhibitor, in Healthy Adults

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Hsp70-derived octapeptide

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  Catalog
Abmole Inhibitor Catalog




Keywords: Icapamespib, PU-HZ151 supplier, HSP, inhibitors, activators

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