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 About 30 results found for searched term "HSP" (0.012 seconds)

Cat.No.  Name Information
M1679 BIIB021 BIIB021 (CNF2024) is an orally available synthetic non-ansamycin Hsp90 inhibitor with ki value of 1.7nM.
M1725 CUDC-305 CUDC-305 is a heat shock protein 90 (HSP90) inhibitor of the novel imidazopyridine class.
M1741 Ganetespib Ganetespib (STA-9090) is a potent synthetic small molecule inhibitor of Hsp90 with potential antineoplastic activity.
M1762 Luminespib (AUY922) Luminespib (AUY922) is a small molecule Heat Shock Protein 90 (HSP90) inhibitor with IC50 values of 13 and 21 nM for HSP90α and HSP90β respectively.
M1798 NVP-HSP990 NVP-HSP990 is an orally bioavailable inhibitor of human heat-shock protein 90 (Hsp90) with potential antineoplastic activity.
M1908 NVP-BEP800 NVP-BEP800 is a novel, fully synthetic, orally bioavailable inhibitor of Hsp90β with an IC50 of 58 nM.
M1949 Onalespib (AT13387) Onalespib (AT13387) is a novel, high-affinity heat-shock protein 90 (HSP90) inhibitor with IC50 of 18 nM in A375 cells.
M2003 PF-04929113 PF-04929113 (SNX-5422) is a potent and selective Hsp90 inhibitor with Kd of 41 nM.
M2070 XL888 XL888 is a novel small-molecule inhibitor of HSP90 with IC50 of 24 nM.
M2320 17-AAG (Tanespimycin) 17-AAG (Tanespimycin) is a potent HSP90 inhibitor with IC50of 5 nM.
M2321 17-DMAG (Alvespimycin) hydrochloride 17-DMAG (Alvespimycin, KOS-1022, NSC 707545) hydrochloride is a potent HSP90 inhibitor with IC50 of 62 nM.
M2776 IPI-493 IPI-493 is a potent and orally bioavailable HSP90 inhibitor with Ki of 21 nM.
M2777 IPI-504 hydrochloride IPI-504 (Retaspimycin) hydrochloride is a potent inhibitor of HSP90 with EC50 of 63 nM.
M2885 NMS-E973 NMS-E973 is a potent and selective Hsp90 inhibitor with DC50 of <10 nM for Hsp90 binding, no activiy against a panel of 52 diverse protein kinases.
M2943 Pifithrin-μ Pifithrin-μ is a specific p53 inhibitor by reducing its affinity to Bcl-xL and Bcl-2, and also inhibits HSP70 function and autophagy.
M3116 VER 155008 VER-155008 is a potent inhibitor of the HSP70 family, with IC50 of 0.5 μM and 2.6 μM for HSP70 and Grp78, respectively, exhibits >100-fold selectivity over HSP90.
M3117 VER-49009 VER-49009 is a potent HSP90 inhibitor with IC50 of 47 nM for HSP90β.
M3197 MPC-3100 MPC-3100 is a fully synthetic and potent Hsp90 inhibitor with IC50 of 60 nM.
M3528 SNX-2112 SNX-2112 selectively binds to the ATP pocket of HSP90α and HSP90β with Ka of 30 nM and 30 nM, uniformly more potent than 17-AAG.
M3561 Geldanamycin Geldanamycin is a natural existing HSP90 inhibitor with Kd of 1.2 μM, specifically disrupts glucocorticoid receptor (GR)/HSP association.
M3563 KW-2478 KW-2478 is a nonansamycin HSP90 inhibitor with IC50 of 3.8 nM.
M3683 Retaspimycin Retaspimycin is a novel, water-soluble, potent inhibitor of heat-shock protein 90 (Hsp90).
M3776 CH5138303 CH5138303 is an orally available Hsp90 inhibitor with Kd of 0.48 nM.
M4618 Eupalinolide A Eupalinolide A, isolated from Eupatorium lindleyanum, induces the expression of HSP70 via the activation of HSF1 by inhibiting the interaction between HSF1 and HSP90.
M4771 Dihydroberberine Dihydroberberine inhibited the human Ether-related gene (hERG) channel and significantly reduced the expression of heat shock protein 90 (Hsp90) and its interaction with hERG. Dihydroberberine has anti-inflammatory, antiatherosclerotic, hylipidemic and antitumor activities.
M6075 HA15 HA15 is a molecule that targets specifically BiP/GRP78/HSPA5. HA15 displays anti-cancerous activity on all melanoma cells tested, including cells isolated from patients and cells that developed resistance to BRAF inhibitors.
M6512 BIX BIX is a biP (Hsp70-5) ER chaperone inducer.
M6571 CCT 018159 CCT 018159 is a hsp90 inhibitor.
M6697 EC 144 EC 144 is a high affinity, potent and selective Hsp90 inhibitor.
M7185 Radicicol Radicicol is a hsp90 inhibitor. Antifungal antibiotic.

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