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CYM 50260

Cat. No. M6642

All AbMole products are for research use only, cannot be used for human consumption.

CYM 50260 Structure

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Quality Control & Documentation
Biological Activity

CYM 50260 is a potent sphingosine-1-phosphate receptor 4 (S1P4) agonist (EC50 = 45 nM). Displays no activity at other S1P receptor subtypes (S1P1-3 and S1P5) at concentrations up to 25 μM.

Chemical Information
Molecular Weight 350.6
Formula C14H11Cl3FNO2
CAS Number 1355026-60-6
Solubility (25°C) DMSO 35.06 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Doherty, et al. J Med Chem. Discovery of potent, orally available vanilloid receptor-1 antagonists Structure-activity relationship of N-aryl cinnamides.

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Keywords: CYM 50260 supplier, S1P Receptor, inhibitors, activators

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