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CK 666

Cat. No. M6611

All AbMole products are for research use only, cannot be used for human consumption.

CK 666 Structure
Size Price Availability Quantity
10mg USD 170  USD170 In stock
50mg USD 650  USD650 In stock
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Quality Control & Documentation
Biological Activity

Ck-666 is a cell-permeable inhibitor (IC50=12 μM) of the Arp2/3 complex, which binds to the Arp2/3 complex and stabilizes the inactive state of the complex, preventing the movement of Arp2 and Arp3 subunits into the active filamentous conformation.

Chemical Information
Molecular Weight 296.34
Formula C18H17FN2O
CAS Number 442633-00-3
Solubility (25°C) DMSO 29.63 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Hill, et al. Bioorg Med Chem Lett. Long chain amines and long chain ammonium salts as novel inhibitors of dynamin GTPase activity.

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  Catalog
Abmole Inhibitor Catalog




Keywords: CK 666 supplier, Actin-Related Protein, inhibitors, activators

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