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CCT251545 is an orally active, potent WNT inhibitor with an IC50 value of 5 nM for WNT inhibition in 7dF3 cells.In addition, CCT251545 is a selective chemical probe for studies related to the roles of CDK8 and CDK19 in human diseases.
| Molecular Weight | 421.92 |
| Formula | C23H24ClN5O |
| CAS Number | 1661839-45-7 |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[3] Thomas G Boyer. Nat Chem Biol. Transcriptional kinases: Less is more (or less)
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