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BMS-779788

Cat. No. M14461

All AbMole products are for research use only, cannot be used for human consumption.

BMS-779788 Structure
Synonym:

EXEL04286652; XL-652; BMS-788

Price and Availability

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Quality Control & Documentation
Biological Activity

BMS-779788 is a LXR partial agonist with IC50 values of 68 nM for LXRα and 14 nM for LXRβ.

Chemical Information
Molecular Weight 509.06
CAS Number 918348-67-1
Solubility (25°C) DMSO 90 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Monica L Adams, et al. Dehydration and Stabilization of a Reactive Tertiary Hydroxyl Group in Solid Oral Dosage Forms of BMS-779788

[2] Todd G Kirchgessner, et al. Pharmacological characterization of a novel liver X receptor agonist with partial LXRα activity and a favorable window in nonhuman primates

[3] Ellen Kick, et al. Liver X receptor (LXR) partial agonists: biaryl pyrazoles and imidazoles displaying a preference for LXRβ

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  Catalog
Abmole Inhibitor Catalog




Keywords: BMS-779788, EXEL04286652; XL-652; BMS-788 supplier, Liver X Receptor, inhibitors, activators

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