Inhibitor/Activator
| Cat.No. | Name | Information |
|---|---|---|
| M53885 | Cortistatin-14 | Cortistatin-14, a neuropeptide have structural similarity to somatostatin-14, binds and exerts its function via the somatostatin receptors (sst1-sst5). |
| M25611 | Cyclosomatostatin acetate | Cyclosomatostatin acetate is a potent somatostatin (SST) receptor antagonist. Cyclosomatostatin acetate can inhibit somatostatin receptor type 1 (SSTR1) signaling and decreases cell proliferation, ALDH+ cell population size and sphere-formation in colorectal cancer (CRC) cells. |
| M20863 | Lanreotide acetate | Lanreotide (Laromustine, Angiopeptin, BIM 23014, Dermopeptin, Ipstyl, ITM-014, Somatulina, Somatuline, Lanreotidum) acetate, an analog of the native somatostatin peptide, is a physiological inhibitor of growth hormone (GH). Lanreotide also has antitumoral effects. |
| M14062 | Octreotide | Octreotide is a somatostatin analog that binds to the somatostatin receptor, mainly subtypes 2, 3, and 5, increases Gi activity, and reduces intracellular cAMP production. |
| M11321 | Angiopeptin TFA | Angiopeptin TFA, a cyclic octapeptide analog of somatostatin, is an SST2 / SST5 receptor partial agonist with IC50 values of 0.26 nM and 6.92 nM, respectively. Angiopeptin TFA inhibits growth hormone release and insulin-like growth factor-1 (IGF-1) production. Angiopeptin TFA inhibits adenylate cyclase or stimulates extracellular acidification. Angiopeptin TFA has the potential to be used in the study of coronary atherosclerosis. |
| M10281 | Somatostatin | Somatostatin is a tetradecapeptide which can suppress the growth hormone (GH) secretion, and regulate the endocrine system to control the pituitary hormone secretion in human CNS. |
| M10248 | Lanreotide | Lanreotide is a somatostatin analogue, acts as an inhibitor of growth hormone (GH). |
| M9463 | FK962 | FK962 is an enhancer of somatostatin release, exerts cognitive-enhancing actions. |
| M5831 | Octreotide Acetate | Octreotide acetate(SMS 201995 acetate) is a long-acting octapeptide with pharmacologic actions mimicking those of the natural hormone somatostatin. |
| M3815 | Pasireotide | Pasireotide is a somatostatin analog with a 40-fold increased affinity to somatostatin receptor 5 compared to other somatostatin analogs. |
| M54292 | TT-232 | TT-232 (CAP-232), a somatostatin derivative, is a peptide SSTR1/SSTR4 agonist. |
| M54122 | Cyclosomatostatin | Cyclosomatostatin is a potent somatostatin (SST) receptor antagonist. |
| M54102 | Somatostatin-28 (1-14) | Somatostatin-28 (1-14) is an N-terminal fragment of the neuropeptide somatostatin-28. |
| M54030 | CH 275 | CH 275 is a peptide analog of somatostatin and binds preferably to somatostatin receptor 1 (sst1) with a Ki of 52 nM. |
| M54002 | CYN 154806 | CYN 154806, a cyclic octapeptide, is a potent and selective somatostatin sst2 receptor antagonist. |
| M52900 | [Tyr1]-Somatostatin-14 | [Tyr1]-Somatostatin-14 could binds to SSTR2. |
| M52899 | (D-Phe5, Cys6, 11, N-Me-D-Trp8)-Somatostatin-14 (5-12) amide | (D-Phe5,Cys6,11,N-Me-D-Trp8)-Somatostatin-14 (5-12) amide is a somatostatin analog with Kds of 0.61, 11.05, 23.5, 1200 and >1000 nM for SSTR5, SSTR3, SSTR2, SSTR1 and SSTR4, respectively. |
| M52898 | [Tyr12] Somatostatin 28 (1-14) | [Tyr12] Somatostatin 28 (1-14) is an analogue of Somatostatin-28 (1-14). |
| M52897 | BIM-23056 TFA | BIM 23056 TFA, a linear octapeptide, is a potent sst3 and sst5 somatostatin receptor antagonist with Ki values of 10.8, 5.7, respectively. |
| M52896 | Satoreotide | Satoreotide (JR11) is a SSTR2 antagonist. |
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