Inhibitor/Activator
Cat.No. | Name | Information |
---|---|---|
M54030 | CH 275 | CH 275 is a peptide analog of somatostatin and binds preferably to somatostatin receptor 1 (sst1) with a Ki of 52 nM. |
M52900 | [Tyr1]-Somatostatin-14 | [Tyr1]-Somatostatin-14 could binds to SSTR2. |
M52899 | (D-Phe5, Cys6, 11, N-Me-D-Trp8)-Somatostatin-14 (5-12) amide | (D-Phe5,Cys6,11,N-Me-D-Trp8)-Somatostatin-14 (5-12) amide is a somatostatin analog with Kds of 0.61, 11.05, 23.5, 1200 and >1000 nM for SSTR5, SSTR3, SSTR2, SSTR1 and SSTR4, respectively. |
M52898 | [Tyr12] Somatostatin 28 (1-14) | [Tyr12] Somatostatin 28 (1-14) is an analogue of Somatostatin-28 (1-14). |
M52897 | BIM-23056 TFA | BIM 23056 TFA, a linear octapeptide, is a potent sst3 and sst5 somatostatin receptor antagonist with Ki values of 10.8, 5.7, respectively. |
M52896 | Satoreotide | Satoreotide (JR11) is a SSTR2 antagonist. |
M52895 | [Nle8] Somatostatin (1-28) | [Nle8] Somatostatin (1-28) is a derivative of somatosttin (1-28) with norleucine replacing methionine in position 8. |
M52894 | Tyr-(D-Dab4, Arg5, D-Trp8)-cyclo-Somatostatin-14 (4-11) | Tyr-(D-Dab4,Arg5,D-Trp8)-cyclo-Somatostatin-14 (4-11) is a somatostatin agonist that can be used in cancer research. |
M52893 | Cortistatin 14, human, rat | Cortistatin 14, human, rat (CST-14, human, rat), a neuropeptide with neuronal depressant and sleep modulating properties, can bind to all five cloned somatostatin receptors (SSTRs) and ghrelin receptor. |
M52892 | Cortistatin-17 (human) | Cortistatin-17 (human) is a somatostatin neuropeptide with potential for studying diseases such as cancer, inflammation, autoimmunity, fibrosis, and pain. |
M52891 | Cortistatin-29 (human) | Cortistatin-29 (human) is a somatostatin neuropeptide with potential for studying diseases such as cancer, inflammation, autoimmunity, fibrosis, and pain. |
M52890 | Octreotide pamoate | Octreotide (SMS 201-995) pamoate is a somatostatin receptor agonist and synthetic octapeptide endogenous somatostatin analogue. |
M52889 | Nendratareotide | Nendratareotide is a somatostatin analogue. |
M52888 | Angiopeptin | Angiopeptin, a cyclic octapeptide analogue of somatostatin, is a weak sst2/sst5 receptor partial agonist with IC50 values of 0.26 nM and 6.92 nM, respectively. |
M52887 | Ilatreotide | Ilatreotide (SDZ CO61), glycated somatostatin derivative, is a highly potent glycated analog of somatostatin with improved oral activity. |
M52886 | BIM-23190 | BIM-23190, a somatostatin analog, a selective SSTR2 and SSTR5 agonist, exhibits Ki values of 0.34 nM and 11.1 nM for SSTR2 and SSTR5, respectively. |
M45207 | SSTR5 antagonist 2 hydrochloride | SSTR5 antagonist 2 hydrochloride is a potent, orally active, selective antagonist of growth hormone-inhibiting hormone (receptor) subtype 5 (SSTR5) for use in studies related to type 2 diabetes. |
M41948 | NODAGA-LM3 | NODAGA-LM3 can be labeled by 68Ga for PET imaging. |
M41947 | NODAGA-LM3 TFA | NODAGA-LM3 TFA can be labeled by 68Ga for PET imaging. |
M41945 | DOTA-JR11 | DOTA-JR11 is a somatostatin receptor 2 (SSTR2)antagonist. |
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