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PERK Protein kinase R (PKR)-like endoplasmic reticulum kinase


Cat.No.  Name Information
M20356 WAY-354896 WAY-354896 is a Dual activator of Protein Kinase R (PKR) and Protein Kinase R-Like Kinase (PERK).
M13716 CCT020312 CCT020312 is a selective EIF2AK3/PERK activator. CCT020312 elicits EIF2A phosphorylation in cells.
M9242 ISRIB ISRIB is a potent and selective PERK inhibitor with IC50 of 5 nM.
M7425 trans-ISRIB trans-ISRIB is a integrated stress response (ISR) inhibitor.
M2996 Salubrinal Salubrinal is a selective inhibitor of eIF2α dephosphorylation and inhibits ER stress-mediated apoptosis with EC50 of ~15 μM.
M2735 GSK2656157 GSK2656157 is an ATP-competitive and highly selective inhibitor of PERK with IC50 of 0.9 nM, 500-fold greater against a panel of 300 kinases.
M2734 GSK2606414 GSK2606414 is an orally available, potent, and selective PERK inhibitor with IC50 of 0.4 nM, displaying at least 100-fold selectivity over the other EIF2AKs assayed.

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