Free shipping on all orders over $ 500

PDK1 3'-phosphoinositide-dependent kinase 1

Cat.No.  Name Information
M9360 Dicoumarol Dicoumarol is an inhibitor of both NAD(P)H:quinone oxidoreductase 1 (NQO1) and PDK1 with IC50s of 0.37 and 19.42 μM, respectively.
M7562 BX517 BX517 is a potent and selective inhibitor of PDK1 with IC50 of 6 nM.
M4832 NVP-BAG956 NVP-BAG956 is a potent, ATP-competitive and selective dual PDK1 and class I PI 3-K inhibitor (IC50 values are 245, 56, 446, 35 and 117 nM for PDK1 and PI 3-K p110 -α, -β, -δ, and -γ respectively).
M2423 AZD7545 AZD7545 is a potent PDHK inhibitor with IC50 of 36.8 nM and 6.4 nM for PDHK1 and PDHK2, respectively.
M2311 BX-912 BX912 is a selective potent PDK1 inhibitor with IC50 of 12 nM.
M2310 BX-795 BX795 is a potent and specific TBK1, IKKε and PDK-1 inhibitor with IC50 of 6 nM, 41 nM and 111 nM, respectively.
M2115 GSK2334470 GSK2334470 is a highly specific and potent inhibitor of PDK1 with IC50 of 10 nM.
M1848 OSU-03012 OSU-03012 is a novel and potent inhibitor of PDK-1 with an IC50 of 5 µM.
M55320 MP7 MP7 (PDK1 inhibitor) is a phosphoinositide-dependent kinase-1 (PDK1) inhibitor.
M43386 PDKtide PDKtide is a biological active peptide.
M28769 PDK1-IN-RS2  PDK1-IN-RS2 is a mimic of peptide docking motif (PIFtide) and is a substrate-selective PDK1 inhibitor with a Kd of 9 μM. PDK1-IN-RS2 suppresses the activation of the downstream kinases S6K1 by PDK1.
M27891 PS47  PS47 is an inactive E-isomer of PS48. PS48 is an activator of PDK1. PS47 can be used as a negative control for PS48.
M20816 PS210 PS210 is a potent activator of PDK1 that binds to the PIF-pocket and allosterically modulates the active site of PDK1.
M20385 WAY-299338 WAY-299338 is a modulator of the Protein Kinase PDK1.
M20367 WAY-298630 WAY-298630 is a PDK1 modulator
M20162 WAY-352098 WAY-352098 is a modulator of the Protein Kinase PDK1

Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2024 AbMole BioScience. All Rights Reserved.