|M9360||Dicoumarol||Dicoumarol is an inhibitor of both NAD(P)H:quinone oxidoreductase 1 (NQO1) and PDK1 with IC50s of 0.37 and 19.42 μM, respectively.|
|M7562||BX517||BX517 is a potent and selective inhibitor of PDK1 with IC50 of 6 nM.|
|M4832||NVP-BAG956||NVP-BAG956 is a potent, ATP-competitive and selective dual PDK1 and class I PI 3-K inhibitor (IC50 values are 245, 56, 446, 35 and 117 nM for PDK1 and PI 3-K p110 -α, -β, -δ, and -γ respectively).|
|M2423||AZD7545||AZD7545 is a potent PDHK inhibitor with IC50 of 36.8 nM and 6.4 nM for PDHK1 and PDHK2, respectively.|
|M2311||BX-912||BX912 is a selective potent PDK1 inhibitor with IC50 of 12 nM.|
|M2310||BX-795||BX795 is a potent and specific TBK1, IKKε and PDK-1 inhibitor with IC50 of 6 nM, 41 nM and 111 nM, respectively.|
|M2115||GSK2334470||GSK2334470 is a highly specific and potent inhibitor of PDK1 with IC50 of 10 nM.|
|M1848||OSU-03012||OSU-03012 is a novel and potent inhibitor of PDK-1 with an IC50 of 5 µM.|
|M28769||PDK1-IN-RS2||PDK1-IN-RS2 is a mimic of peptide docking motif (PIFtide) and is a substrate-selective PDK1 inhibitor with a Kd of 9 μM. PDK1-IN-RS2 suppresses the activation of the downstream kinases S6K1 by PDK1.|
|M27891||PS47||PS47 is an inactive E-isomer of PS48. PS48 is an activator of PDK1. PS47 can be used as a negative control for PS48.|
|M20816||PS210||PS210 is a potent activator of PDK1 that binds to the PIF-pocket and allosterically modulates the active site of PDK1.|
|M20385||WAY-299338||WAY-299338 is a modulator of the Protein Kinase PDK1.|
|M20367||WAY-298630||WAY-298630 is a PDK1 modulator|
|M20162||WAY-352098||WAY-352098 is a modulator of the Protein Kinase PDK1|
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