| Cat.No. | Name | Information |
|---|---|---|
| M2167 | (+)-JQ1 | (+)-JQ1 is a BET bromodomain inhibitor that acts on BRD4(2) with an IC50 of 33 nM and binds to all bromodomain domains in the BET family, but not to bromodomain domains outside the BET family. JQ1 down-regulates CD47 expression through a C-MYC-mediated pathway, and JQ1 down-regulates CD47 expression through a C-MYC-mediated pathway. |
| M6118 | 666-15 | 666-15 is a potent and selective CREB inhibitor with an IC50 of 81 nM. |
| M2096 | GSK1210151A | GSK1210151A (I-BET151) is an inhibitor of the BET family with IC50 of 0.5 μM, 0.25 μM and 0.79 μM for BRD2, BRD3 and BRD4, respectively. |
| M2903 | OTX015 (Birabresib) | OTX015 is a potent BET bromodomain inhibitor with EC50 ranging from 10 to 19 nM for BRD2, BRD3, and BRD4. |
| M2190 | I-BET-762 | I-BET-762 (GSK525762) is a selective small molecule BET inhibitor. |
| M7126 | PF CBP1 | PF CBP1 is a selective CBP/p300 bromodomain inhibitor. |
| M41667 | BRD4-IN-4 | BRD4-IN-4 is a BRD4 inhibitor (IC50=6.83 μM). |
| M41666 | WWL0245 | WWL0245 is a potent and seletive BRD4 PROTAC. |
| M41665 | TMX1 | TMX1 is a BRD4 covalent molecular glue degrader. |
| M41664 | SJ1461 | SJ1461 is a potent and orally active BET inhibitor. |
| M41663 | BRD4 Inhibitor-28 | BRD4 Inhibitor-28 is an orally active BRD4 Inhibitor. |
| M41662 | IV-275 | IV-275 is an inhibitor of both BRG1 and BRM bromodomains. |
| M41661 | BET bromodomain inhibitor 3 | BET bromodomain inhibitor 3 is BET bromodomain inhibitor. |
| M41660 | CBP-IN-1 | CBP-IN-1 is a potent CBP inhibitor, with an IC50 of 1.5 nM. |
| M41659 | PROTAC BRD4 Degrader-21 | PROTAC BRD4 Degrader-21 is a PROTAC degrader of BRD4. |
| M41658 | BET-IN-14 | BET-IN-14 is an orally active pan BET inhibitor (IC50: 5.35 nM). |
| M41657 | VinSpinIn | VinSpinIn is a Spindlin1 inhibitor (KD: 9.9 nM for SPIN149-262). |
| M41656 | IV-255 | IV-255 is a selective small molecule inhibitor of the BRG1 bromodomain. |
| M41655 | BET BD2-IN-1 | BET BD2-IN-1 is a potent and selective inhibitor of BET BD2 (IC50=1.6 nM). |
| M41654 | SMD-3040 | SMD-3040 is a potent and selective of SMARCA2 PROTAC degrader (DC50: 12 nM). |
| M41653 | PROTAC BRD4 Degrader-20 | PROTAC BRD4 Degrader-20 is an bifunctional compound and an degrader of BRD4. |
| M41652 | GSK737 | GSK737 is a BRD4 BD1 and BD2 inhibitor, with pIC50 values of 5.3 and 7.3 respectively. |
| M41651 | GXF-111 | GXF-111, a PROTAC molecule, can promote selective degradation of cellular BRD3 and BRD4-L. |
| M41650 | BRD4 Inhibitor-27 | BRD4 Inhibitor-27 is a BRD4 inhibitor with IC50 of 9.6 and 11.3 μM for BRD4 BD1 and BRD4 BD2, respectively. |
| M41649 | TRIM24/BRPF1-IN-2 | TRIM24/BRPF1-IN-2 is a potent TRIM24/BRPF1 dual inhibitor, with IC50 values of 0.98 and 1.16 μM, respectively. |
| M41648 | BRD7-IN-2 | BRD7-IN-2 is a potent inhibitor of bromodomain-containing protein 7 (BRD7), targeting to prostate cancer cells. |
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