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DS17701585

Cat. No. M45236

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DS17701585 Structure

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Quality Control & Documentation
Biological Activity

DS17701585 is a selective, orally active inhibitor of EP300 and CBP with IC50 values of 0.040, 0.15, 0.45, and 0.70 µM for CBP, EP300, H3K27, and SOX2, respectively.CAS 번호128-52-56-5

Chemical Information
Molecular Weight 482.55
Formula C24H26N4O5S
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Ryutaro Kanada, et al. Bioorg Med Chem Lett. Discovery of EP300/CBP histone acetyltransferase inhibitors through scaffold hopping of 1,4-oxazepane ring

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  Catalog
Abmole Inhibitor Catalog




Keywords: DS17701585 supplier, Epigenetic Reader Domain, inhibitors, activators

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