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Bradykinin Receptor Bradykinin Receptor

Cat.No.  Name Information
M13916 Icatibant Icatibant (HOE-140) is a potent and specific peptide antagonist of bradykinin B2 receptor with IC50 and Ki of 1.07 nM and 0.798 nM respectively.
M13915 Bradykinin Bradykinin (bradykinin) is a vasodilator active peptide produced by the kinin-releasing enzyme-kinin system that modulates inflammation by causing vasodilation, increasing vascular permeability, and stimulating prostaglandin synthesis.
M10164 Icatibant (HOE 140) acetate Icatibant (HOE-140) acetate is a potent and specific peptide antagonist of bradykinin B2 receptor, with IC50 value of 1.07 nM and Ki value of 0.798 nM, respectively.
M7534 SSR240612 Treatment with the kinin B1 receptor antagonist, SSR240612, provided a protective effect against organ damage by interfering with multiple target functions, including the suppression of B1R-induced inflammation and platelet aggregation.
M3947 ELN 441958 ELN-441958 is a potent, neutral, competitive and selective oral bioavailable bradykinin B1 receptor antagonist with a Ki of 0.26 nM against native human bradykinin B1 receptor.
M54281 [Hyp3]-Bradykinin [Hyp3]-Bradykinin, naturally occurring peptide hormone, is a bradykinin receptor agonist.
M54238 Bradykinin (1-6) Bradykinin (1-6) is an amino-truncated Bradykinin peptide.
M54164 Lys-[Des-Arg9]Bradykinin TFA Lys-[Des-Arg9]Bradykinin TFA, a naturally occurring kinin, is a potent and highly selective bradykinin B1 receptor agonist with a Ki of 0.12 nM, 1.7 nM and 0.23 nM for human, mouse and rabbit B1 receptors, respectively.
M54123 Lobradimil Lobradimil (RMP 7), a synthetic bradykinin analog, is a potent and selective bradykinin B2 receptor agonist (Ki: 0.54 nM).
M54078 [Tyr8] Bradykinin [Tyr8] Bradykinin is a B2 kinin receptor agonist.
M53931 Bradykinin (1-7) Bradykinin (1-7) is an amino-truncated Bradykinin peptide.
M53889 [Des-Arg9]-Bradykinin acetate [Des-Arg9]-Bradykinin acetate is a Bradykinin B1 receptor agonist that displays selectivity for B1 over B2 receptors.
M53707 Bradykinin (1-5) Bradykinin (1-5) is a major stable metabolite of Bradykinin, formed by the proteolytic action of angiotensin-converting enzyme (ACE).
M53249 Methionyl-Lysyl-Bradykinin Methionyl-Lysyl-Bradykinin (Met-Lys-Bradykinin), a Bradykinin analogue, is a kinin.
M53248 Lys-[Des-Arg9]Bradykinin Lys-[Des-Arg9]Bradykinin, a naturally occurring kinin, is a potent and highly selective bradykinin B1 receptor agonist with a Ki of 0.12 nM, 1.7 nM and 0.23 nM for human, mouse and rabbit B1 receptors, respectively.
M53247 Bradykinin (2-9) Bradykinin (2-9) is an amino-truncated Bradykinin peptide.
M53246 [Des-Arg9]-Bradykinin [Des-Arg9]-Bradykinin is a Bradykinin (B1) receptor agonist that displays selectivity for B1 over B2 receptors.
M53245 [Phe8Ψ(CH-NH)Arg9]-Bradykinin [Phe8Ψ(CH-NH)Arg9]-Bradykinin is a selective Bradykinin receptor B2 agonist (not cleaved by protein kinase I/II).
M53244 Des-Arg9-[Leu8]-Bradykinin acetate Des-Arg9-[Leu8]-Bradykinin acetate is potent bradykinin receptor 1 (B1R) antagonist.
M53243 Sar-[D-Phe8]-des-Arg9-Bradykinin Sar-[D-Phe8]-des-Arg9-Bradykinin is a agonist of B1 receptor.




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