Cat.No. | Name | Information |
---|---|---|
M53246 | [Des-Arg9]-Bradykinin | [Des-Arg9]-Bradykinin is a Bradykinin (B1) receptor agonist that displays selectivity for B1 over B2 receptors. |
M13916 | Icatibant | Icatibant (HOE-140) is a potent and specific peptide antagonist of bradykinin B2 receptor with IC50 and Ki of 1.07 nM and 0.798 nM respectively. |
M13915 | Bradykinin | Bradykinin (bradykinin) is a vasodilator active peptide produced by the kinin-releasing enzyme-kinin system that modulates inflammation by causing vasodilation, increasing vascular permeability, and stimulating prostaglandin synthesis. |
M10164 | Icatibant (HOE 140) acetate | Icatibant (HOE-140) acetate is a potent and specific peptide antagonist of bradykinin B2 receptor, with IC50 value of 1.07 nM and Ki value of 0.798 nM, respectively. |
M7534 | SSR240612 | Treatment with the kinin B1 receptor antagonist, SSR240612, provided a protective effect against organ damage by interfering with multiple target functions, including the suppression of B1R-induced inflammation and platelet aggregation. |
M3947 | ELN 441958 | ELN-441958 is a potent, neutral, competitive and selective oral bioavailable bradykinin B1 receptor antagonist with a Ki of 0.26 nM against native human bradykinin B1 receptor. |
M54281 | [Hyp3]-Bradykinin | [Hyp3]-Bradykinin, naturally occurring peptide hormone, is a bradykinin receptor agonist. |
M54238 | Bradykinin (1-6) | Bradykinin (1-6) is an amino-truncated Bradykinin peptide. |
M54164 | Lys-[Des-Arg9]Bradykinin TFA | Lys-[Des-Arg9]Bradykinin TFA, a naturally occurring kinin, is a potent and highly selective bradykinin B1 receptor agonist with a Ki of 0.12 nM, 1.7 nM and 0.23 nM for human, mouse and rabbit B1 receptors, respectively. |
M54123 | Lobradimil | Lobradimil (RMP 7), a synthetic bradykinin analog, is a potent and selective bradykinin B2 receptor agonist (Ki: 0.54 nM). |
M54078 | [Tyr8] Bradykinin | [Tyr8] Bradykinin is a B2 kinin receptor agonist. |
M53931 | Bradykinin (1-7) | Bradykinin (1-7) is an amino-truncated Bradykinin peptide. |
M53889 | [Des-Arg9]-Bradykinin acetate | [Des-Arg9]-Bradykinin acetate is a Bradykinin B1 receptor agonist that displays selectivity for B1 over B2 receptors. |
M53707 | Bradykinin (1-5) | Bradykinin (1-5) is a major stable metabolite of Bradykinin, formed by the proteolytic action of angiotensin-converting enzyme (ACE). |
M53249 | Methionyl-Lysyl-Bradykinin | Methionyl-Lysyl-Bradykinin (Met-Lys-Bradykinin), a Bradykinin analogue, is a kinin. |
M53248 | Lys-[Des-Arg9]Bradykinin | Lys-[Des-Arg9]Bradykinin, a naturally occurring kinin, is a potent and highly selective bradykinin B1 receptor agonist with a Ki of 0.12 nM, 1.7 nM and 0.23 nM for human, mouse and rabbit B1 receptors, respectively. |
M53247 | Bradykinin (2-9) | Bradykinin (2-9) is an amino-truncated Bradykinin peptide. |
M53245 | [Phe8Ψ(CH-NH)Arg9]-Bradykinin | [Phe8Ψ(CH-NH)Arg9]-Bradykinin is a selective Bradykinin receptor B2 agonist (not cleaved by protein kinase I/II). |
M53244 | Des-Arg9-[Leu8]-Bradykinin acetate | Des-Arg9-[Leu8]-Bradykinin acetate is potent bradykinin receptor 1 (B1R) antagonist. |
M53243 | Sar-[D-Phe8]-des-Arg9-Bradykinin | Sar-[D-Phe8]-des-Arg9-Bradykinin is a agonist of B1 receptor. |
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