| Cat.No. | Name | Information |
|---|---|---|
| M10146 | TRV-120027 TFA | TRV-120027 (also known as TRV027) is an angiotensin II receptor type 1 (AT1R) antagonist and engages ß-arrestins while blocking G-protein signaling. |
| M9079 | Angiotensin-(1-7) | Angiotensin (1-7) is a synthetic heptapeptide identical to endogenous angiotensin-(1-7), inhibits purified canine angiotensin converting enzyme (ACE) activity with an IC50 of 0.65 μM. |
| M5731 | LCZ696 | LCZ696, consisting of Valsartan and Sacubitril in a 1:1 molar ratio, is a first-in-class dual-action angiotensin receptor-neprilysin inhibitor (ARNi,angiotensin receptor-neprilysin inhibitor) for the study of hypertension and heart failure. |
| M3507 | Valsartan | Valsartan is an angiotensin II receptor antagonist with IC50 of ranging from 39.5 to 116 μM. |
| M2106 | Azilsartan | Azilsartan (TAK-536) is an angiotensin II type 1 (AT1) receptor antagonist with IC50 of 2.6 nM. Azilsartan induces ROS formation and apoptosis in HepG2 cells. Azilsartan shows neuroprotective and anticancer activity. |
| M54314 | TRV055 | TRV055, a G-protein-biased agonist, is a Gq-biased ligand of the angiotensin II receptor type 1 (AT1R). |
| M54072 | TRV056 | TRV056 is a Gq-biased ligand of the angiotensin II receptor type 1 (AT1R). TRV056 is efficacious in stimulating cellular Gq-mediated signaling. TRV056 can be used to develop the Gq-biased AT1R agonists. |
| M45381 | Angiotensin III, human, mouse | Angiotensin III, human, mouse is a heptapeptide and an angiotensin type 2 receptor (AT2R) agonist with IC50 values of 0.648 nM and 21.1 nM for AT2R and AT1R, respectively. |
| M45380 | Saralasin TFA | Saralasin TFA is an octapeptide analog of Angiotensin II and a competitive angiotensin II receptor antagonist with a Ki value of 0.32 nM (74% of binding sites) and partial agonist activity. It has a Ki value of 0.32 nM (74% of binding sites) and partial agonist activity. It can be used in studies related to renal vascular hypertension and renin-dependent (angiotensinogenic) hypertension. |
| M13910 | Eprosartan | Eprosartan (SKF-108566J free base) is a selective, competitive, nonpeptid and orally active angiotensin II receptor antagonist, used as an antihypertensive. |
| M13909 | CGP-42112 | CGP-42112 (CGP-42112A) is a potent Angiotensin-II subtype 2 receptor(AT2 R) agonist. |
| M13908 | AVE 0991 sodium salt | AVE 0991 sodium salt is a nonpeptide and orally active Ang-(1-7) receptor Mas agonist. AVE 0991 competes for high-affinity binding of [125I]-Ang-(1-7) to bovine aortic endothelial cell membranes with IC50 of 21 nM. |
| M13907 | AT2 receptor agonist C21 | AT2 receptor agonist C21 is a druglike selective angiotensin II AT2 receptor agonist with Ki values of 0.4 nM and >10 µM for the AT2 receptor and AT1 receptor, respectively. |
| M13906 | Angiotensin II human TFA | Angiotensin II human (Angiotensin II) TFA is a vasoconstrictor and a major bioactive peptide of the renin/angiotensin system. |
| M13905 | Angiotensin II human acetate | Angiotensin II human (Angiotensin II) acetate is a vasoconstrictor and a major bioactive peptide of the renin/angiotensin system. |
| M13904 | Angiotensin (1-7) (acetate) | Angiotensin 1-7 (Ang-(1-7)) acetate is an endogenous heptapeptide from the renin-angiotensin system (RAS) with a cardioprotective role due to its anti-inflammatory and anti-fibrotic activities in cardiac cells. |
| M10358 | C-Type Natriuretic Peptide (CNP) (1-22), human | C-Type Natriuretic Peptide (CNP) (1-22), human is the 1-22 fragment of C-Type Natriuretic Peptide. |
| M10273 | AVE 0991 | AVE 0991 is an orally active agonist of angiotensin-(1-7) receptor with IC50 of 21 nM. |
| M9852 | BIBS39 | BIBS39 is a new nonpeptide angiotensin II (AII) receptor antagonist. |
| M9091 | A-779 | A-779 is a specific antagonist of G-protein coupled receptor (Mas receptor). |
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