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Androgen Receptor Androgen Receptor

Inhibitors

Cat.No.  Name Information
M1973 Ostarine (GTx-024) Ostarine (GTx-024 and MK-2866) is an investigational selective androgen receptor modulator (SARM) with Ki of 3.8 nM.
M6033 Dihydrotestosterone Dihydrotestosterone is an androgen (male hormone). Specifically it's the strongest of the androgens.
M6105 Testosterone Testosterone is an androgen, which binds the androgen receptor.
M5565 Dexmedetomidine HCl Dexmedetomidine Hydrochloride is an agonist of adrenergic alpha-2 receptor, which is used in veterinary medicine for its analgesic and sedative properties.
M20966 Ligandrol (LGD-4033, VK-5211) Ligandrol (LGD-4033, VK-5211) is a novel nonsteroidal, oral selective androgen receptor modulator with high affinity (Ki of ∼1 nM) and selectivity.
M20065 WAY-298516 WAY-298516 is a modulating rad51
M14623 UT-155 UT-155 is a selective and potent androgen receptor (AR) antagonist, with a Ki of 267 nM for UT-155 binding to AR-LBD.
M14622 Stanolone benzoate Stanolone benzoate (Androstanolone benzoate) is a synthetic androgen and anabolic steroid.
M14621 S-23 S-23 is an orally active selective androgen receptor modulator (SARM) with a Ki of 1.7 nM.
M14620 Vosilasarm Vosilasarm (RAD140) is a potent, orally active, nonsteroidal selective androgen receptor modulator (SARM) with a Ki of 7 nM. Vosilasarm shows good selectivity over other steroid hormone nuclear receptors.
M14619 MK-0773 MK-0773 is a selective androgen receptor modulators (SARMs) that binds to AR with an IC50 of 6.6 nM.
M14618 LY2452473 LY2452473 is an orally bioavailable, selective androgen receptor modulator (SARM).
M14617 GLPG0492 GLPG0492 is a non-steroidal selective androgen receptor modulator (potency 12 nM). GLPG0492 has the potential for the research of musculo-skeletal diseases such as sarcopenia and cachexia.
M14616 Dehydroisoandrosterone 3-acetate Dehydroepiandrosterone 3-acetate is a testosterone/estrogen precursor and known modulator of vertebrate aggression.
M14615 BMS-564929 BMS-564929 is an androgen receptor (AR) agonist, binds to androgen receptor (AR) with a Ki of 2.11±0.16 nM.
M14614 ACP-105 ACP-105 is an orally available, selective amd potent androgen receptor modulator (SARM), with pEC50s of 9.0 and 9.3 for AR wild type and T877A mutant, respectively.
M14613 3,3'-Diindolylmethane 3,3'-Diindolylmethane is a strong, pure androgen receptor (AR) antagonist.
M11350 Triptophenolide Triptophenolide is a colorless crystal isolated from the ethyl acetate extract of Triptophenolide.
M10965 ORM-15341 ORM-15341 is a potent androgen receptor (AR) antagonist that acts on AR-HEK293 cells with an IC50 value of 38 nM.
M10960 Ralaniten Ralaniten (EPI-002) is an effective and orally active androgen receptor N-terminal domain (AR-NTD) antagonist. Ralaniten inhibits AR transcriptional activity,IC50 The value is 7.4 μM. Ralanites can be used in the study of castration-resistant prostate cancer (CRPC).
M10958 JNJ-63576253 JNJ-63576253 (TRC-253) is a potent and orally active complete antagonist of the androgen receptor against F877L mutant AR and wild-type AR in LNCaP cells IC50 The values are 37 and 54 nM, respectively. JNJ-63576253 can be used in the study of castration-resistant prostate cancer (CRPC).
M10306 Bavdegalutamide (ARV-110) Bavdegalutamide (ARV-110) is an oral, specific androgen receptor (AR) PROTAC degrader.
M9956 Darolutamide Darolutamide (ODM-201) is a new-generation, potent and selective androgen receptor (AR) inhibitor.
M9149 MI-136 MI-136 inhibits DHT-induced expression of androgen receptor (AR) target genes.



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