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Inhibitors
| Cat.No. | Name | Information |
|---|---|---|
| M10306 | Bavdegalutamide (ARV-110) | Bavdegalutamide (ARV-110) is an oral, specific androgen receptor (AR) PROTAC degrader. |
| M9956 | Darolutamide | Darolutamide (ODM-201) is a new-generation, potent and selective androgen receptor (AR) inhibitor. |
| M9149 | MI-136 | MI-136 inhibits DHT-induced expression of androgen receptor (AR) target genes. |
| M9061 | Dehydroepiandrosterone | Dehydroepiandrosterone is an effective antiapoptotic factor. |
| M8908 | ASC-J9 | ASC-J9, also known as GO-Y025 and Dimethylcurcumin, suppressesing castration-resistant prostate cancer growth through degradation of full-length and splice variant androgen receptors. |
| M8128 | R1881 | R1881 (Metribolone) is an orally active, non-aromatisable androgen and anabolic steroid. |
| M7561 | GSK-2881078 | GSK 2881078 is a selective androgen receptor modulator potentially for the treatment of cachexia. GSK 2881078 is a selective androgen receptor modulator (SARM) that is being evaluated for effects on muscle growth and strength in subjects with muscle wasting to improve their physical function. |
| M6269 | Indacaterol | Indacaterol(Onbrez; Arcapta) is an ultra-long-acting β-adrenoceptor agonist. |
| M6123 | Nandrolone phenylpropionate | Nandrolone phenylpropionate (NPP) is an anabolic-androgenic steroid. The low androgenicity and enhanced anabolic activity of NPP has shown to positively influence calcium metabolism and to increase bone mass in osteoporosis. |
| M6122 | ChlordehydroMethyl Testosterone | Testosterone is normally present in the circulation of both men and women. Due to the dynamic regulation of endogenous testosterone production, including the acute effects of competition and exercise, testosterone concentrations may vary considerably within and among individuals. |
| M6121 | Testosterone phenylpropionate | Testosterone phenylpropionate is a synthetic anabolic-androgenic steroid (AAS) and an androgen ester. |
| M6120 | Testosterone isocaproate | Testosterone Isocaproate help in increasing the body weight and will also help in gaining the strength and also help in losing fat in the body and gives an increase in libido, red blood cells, stamina and quick recovery after heavy training. |
| M6119 | Testosterone Enanthate | Androcur-treatment abolished testosterone-reduced cAMP, coupled with a changed expressional milieu of cAMP signaling elements. Results from in vitro experiments suggest that some of these effects are testosterone-AR dependent, while others could be due to disturbed LH and/or other signals. |
| M6117 | Testosterone decanoate | As with all forms of testosterone,Testosterone Decanoate will cause weight and strength gain, fat loss, a libido increase, an increase in IGF-1 levels, Red Blood Cell count, and of course increased recovery from training |
| M6116 | Drostanolone Enanthate | Drostanolone is one of the most frequently detected anabolic androgenic steroids in doping control analysis. |
| M6114 | Metandienone | Metandienone is a synthetic anabolic steroid that is prohibited in sports by the World Anti-Doping Agency (WADA). |
| M6106 | 17α-Methyltestosterone | 17α-Methyltestosterone has similar binding affinity to AR and similar androgenic and anabolic activities as testosterone. IC50 value: 17 nM (Ki) Target:Androgen Receptor. |
| M6105 | Testosterone | Testosterone is an androgen, which binds the androgen receptor. |
| M6099 | Boldenone Undecylenate | Boldenone undecylenate(Equipoise) is a synthetic steroid which has a similar effect as the natural steroid testosterone. |
| M6033 | Dihydrotestosterone | Dihydrotestosterone is an androgen (male hormone). Specifically it's the strongest of the androgens. |
| M6028 | Trenbolone acetate | Trenbolone acetate (TBA; RU1697; Finaplix) is a synthetic androgen steroid with anabolic properties. |
| M6004 | Testosterone propionate | Testosterone Propionate is an efficient androgenic hormone for the treatment of low testosterone. |
| M5659 | Flutamide | Flutamide is an antiandrogen drug, with its active metablolite binding at androgen receptor with Ki values of 55 nM, and primarily used to treat prostate cancer. |
| M5657 | Fluoxymesterone | Fluoxymesterone is an Androgen. The mechanism of action of fluoxymesterone is as an Androgen Receptor Agonist. |
| M5586 | DL-Epinephrine | DL-Epinephrine(DL-Adrenaline) is a hormone and a neurotransmitter. |
| M5565 | Dexmedetomidine HCl | Dexmedetomidine Hydrochloride is an agonist of adrenergic alpha-2 receptor, which is used in veterinary medicine for its analgesic and sedative properties. |
| M5544 | Cyproterone Acetate | Cyproterone acetate is an androgen receptor (AR) antagonist with IC50 of 7.1 nM, as well as a weak progesterone receptor agonist with weak pro-gestational and glucocorticoid activity. |
| M5454 | Betaxolol HCl | Betaxolol is a β1 adrenergic receptor blocker with IC50 of 6 μM. |
| M5396 | Alfuzosin HCl | Alfuzosin HCl is an alpha1 receptor antagonist used to treat benign prostatic hyperplasia (BPH). |
| M5395 | Alfuzosin | Alfuzosin is an α1 adrenergic receptor antagonist used to treat benign prostatic hyperplasia (BPH). |
| M5035 | 17 alpha-propionate | 17 alpha-propionate is a new topical and peripherally selective androgen antagonist. |
| M3750 | TAK-700 | TAK-700 (Orteronel) is an investigational, oral, nonsteroidal, selective, reversible inhibitor of 17,20-lyase, a key enzyme in the production of androgenic hormones. |
| M3685 | Mesterolone | The Mesterolone is an orally applicable androgen, and DHT derivative. |
| M3502 | Testosterone cypionate | Testosterone cypionate is the oil-soluble 17 (beta)-cyclopentylpropionate ester of the androgenic hormone testosterone. |
| M3459 | Lubiprostone | Lubiprostone is a gastrointestinal agent used for the treatment of idiopathic chronic constipation. |
| M3234 | (R)-Bicalutamide | (R)-Bicalutamide is an active competitive non-steroidal androgen receptor antagonist with an IC50 of 0.17 μM for MDA 453 cells. |
| M3191 | Nilutamide | Nilutamide (RU 23908) is an androgen receptor (AR) blocker with IC50 of 0.4 μM. |
| M3028 | Spironolactone | Spironolactone is a potent antagonist of the androgen receptor with IC50 of 77 nM. |
| M2717 | Galeterone | Galeterone is a selective CYP17 inhibitor and androgen receptor (AR) antagonist with IC50 of 300 nM and 384 nM, respectively, and is a potent inhibitor of human prostate tumor growth. |
| M2670 | Epiandrosterone | Epiandrosterone is a steroid hormone with weak androgenic activity, is a natural metabolite of DHEA. |
| M2344 | RU 58841 | RU 58841 is a specific androgen receptor antagonist or anti-androgen. |
| M2270 | Apalutamide (ARN-509) | Apalutamide (ARN-509) is a novel androgen receptor (AR) antagonist for the treatment of castration-resistant prostate cancer (CRPC). |
| M2092 | AZD3514 | AZD3514 is a potent, small-molecule androgen receptor downregulator with potential anticancer cancer activity. |
| M1986 | Andarine | Andarine (GTx-007, S-4) is an orally active partial agonist for androgen receptors. |
| M1973 | Ostarine (GTx-024) | Ostarine (GTx-024 and MK-2866) is an investigational selective androgen receptor modulator (SARM) with Ki of 3.8 nM. |
| M1960 | Bicalutamide | Bicalutamide is an orally active non-steroidal androgen receptor antagonist (IC50 = 190 nM). |
| M1839 | MDV3100 | MDV3100 is an orally bioavailable, organic, non-steroidal small molecule targeting the androgen receptor (AR) with potential antineoplastic activity. |
| M1586 | Norelgestromin | Norgestimate and its metabolite norelgestromin possess weak androgen-like properties. |
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