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Abmole Inhibitor Catalog 2017

Androgen Receptor Androgen Receptor


Cat.No.  Name Information
M10306 Bavdegalutamide (ARV-110) Bavdegalutamide (ARV-110) is an oral, specific androgen receptor (AR) PROTAC degrader.
M9956 Darolutamide Darolutamide (ODM-201) is a new-generation, potent and selective androgen receptor (AR) inhibitor.
M9149 MI-136 MI-136 inhibits DHT-induced expression of androgen receptor (AR) target genes.
M9061 Dehydroepiandrosterone Dehydroepiandrosterone is an effective antiapoptotic factor.
M8908 ASC-J9 ASC-J9, also known as GO-Y025 and Dimethylcurcumin, suppressesing castration-resistant prostate cancer growth through degradation of full-length and splice variant androgen receptors.
M8128 R1881 R1881 (Metribolone) is an orally active, non-aromatisable androgen and anabolic steroid.
M7561 GSK-2881078 GSK 2881078 is a selective androgen receptor modulator potentially for the treatment of cachexia. GSK 2881078 is a selective androgen receptor modulator (SARM) that is being evaluated for effects on muscle growth and strength in subjects with muscle wasting to improve their physical function.
M6269 Indacaterol Indacaterol(Onbrez; Arcapta) is an ultra-long-acting β-adrenoceptor agonist.
M6123 Nandrolone phenylpropionate Nandrolone phenylpropionate (NPP) is an anabolic-androgenic steroid. The low androgenicity and enhanced anabolic activity of NPP has shown to positively influence calcium metabolism and to increase bone mass in osteoporosis.
M6122 ChlordehydroMethyl Testosterone Testosterone is normally present in the circulation of both men and women. Due to the dynamic regulation of endogenous testosterone production, including the acute effects of competition and exercise, testosterone concentrations may vary considerably within and among individuals.
M6121 Testosterone phenylpropionate Testosterone phenylpropionate is a synthetic anabolic-androgenic steroid (AAS) and an androgen ester.
M6120 Testosterone isocaproate Testosterone Isocaproate help in increasing the body weight and will also help in gaining the strength and also help in losing fat in the body and gives an increase in libido, red blood cells, stamina and quick recovery after heavy training.
M6119 Testosterone Enanthate Androcur-treatment abolished testosterone-reduced cAMP, coupled with a changed expressional milieu of cAMP signaling elements. Results from in vitro experiments suggest that some of these effects are testosterone-AR dependent, while others could be due to disturbed LH and/or other signals.
M6117 Testosterone decanoate As with all forms of testosterone,Testosterone Decanoate will cause weight and strength gain, fat loss, a libido increase, an increase in IGF-1 levels, Red Blood Cell count, and of course increased recovery from training
M6116 Drostanolone Enanthate Drostanolone is one of the most frequently detected anabolic androgenic steroids in doping control analysis.
M6114 Metandienone Metandienone is a synthetic anabolic steroid that is prohibited in sports by the World Anti-Doping Agency (WADA).
M6106 17α-Methyltestosterone 17α-Methyltestosterone has similar binding affinity to AR and similar androgenic and anabolic activities as testosterone. IC50 value: 17 nM (Ki) Target:Androgen Receptor.
M6105 Testosterone Testosterone is an androgen, which binds the androgen receptor.
M6099 Boldenone Undecylenate Boldenone undecylenate(Equipoise) is a synthetic steroid which has a similar effect as the natural steroid testosterone.
M6033 Dihydrotestosterone Dihydrotestosterone is an androgen (male hormone). Specifically it's the strongest of the androgens.
M6028 Trenbolone acetate Trenbolone acetate (TBA; RU1697; Finaplix) is a synthetic androgen steroid with anabolic properties.
M6004 Testosterone propionate Testosterone Propionate is an efficient androgenic hormone for the treatment of low testosterone.
M5659 Flutamide Flutamide is an antiandrogen drug, with its active metablolite binding at androgen receptor with Ki values of 55 nM, and primarily used to treat prostate cancer.
M5657 Fluoxymesterone Fluoxymesterone is an Androgen. The mechanism of action of fluoxymesterone is as an Androgen Receptor Agonist.
M5586 DL-Epinephrine DL-Epinephrine(DL-Adrenaline) is a hormone and a neurotransmitter.
M5565 Dexmedetomidine HCl Dexmedetomidine Hydrochloride is an agonist of adrenergic alpha-2 receptor, which is used in veterinary medicine for its analgesic and sedative properties.
M5544 Cyproterone Acetate Cyproterone acetate is an androgen receptor (AR) antagonist with IC50 of 7.1 nM, as well as a weak progesterone receptor agonist with weak pro-gestational and glucocorticoid activity.
M5454 Betaxolol HCl Betaxolol is a β1 adrenergic receptor blocker with IC50 of 6 μM.
M5396 Alfuzosin HCl Alfuzosin HCl is an alpha1 receptor antagonist used to treat benign prostatic hyperplasia (BPH).
M5395 Alfuzosin Alfuzosin is an α1 adrenergic receptor antagonist used to treat benign prostatic hyperplasia (BPH).
M5035 17 alpha-propionate 17 alpha-propionate is a new topical and peripherally selective androgen antagonist.
M3750 TAK-700 TAK-700 (Orteronel) is an investigational, oral, nonsteroidal, selective, reversible inhibitor of 17,20-lyase, a key enzyme in the production of androgenic hormones.
M3685 Mesterolone The Mesterolone is an orally applicable androgen, and DHT derivative.
M3502 Testosterone cypionate Testosterone cypionate is the oil-soluble 17 (beta)-cyclopentylpropionate ester of the androgenic hormone testosterone.
M3459 Lubiprostone Lubiprostone is a gastrointestinal agent used for the treatment of idiopathic chronic constipation.
M3234 (R)-Bicalutamide (R)-Bicalutamide is an active competitive non-steroidal androgen receptor antagonist with an IC50 of 0.17 μM for MDA 453 cells.
M3191 Nilutamide Nilutamide (RU 23908) is an androgen receptor (AR) blocker with IC50 of 0.4 μM.
M3028 Spironolactone Spironolactone is a potent antagonist of the androgen receptor with IC50 of 77 nM.
M2717 Galeterone Galeterone is a selective CYP17 inhibitor and androgen receptor (AR) antagonist with IC50 of 300 nM and 384 nM, respectively, and is a potent inhibitor of human prostate tumor growth.
M2670 Epiandrosterone Epiandrosterone is a steroid hormone with weak androgenic activity, is a natural metabolite of DHEA.
M2344 RU 58841 RU 58841 is a specific androgen receptor antagonist or anti-androgen.
M2270 Apalutamide (ARN-509) Apalutamide (ARN-509) is a novel androgen receptor (AR) antagonist for the treatment of castration-resistant prostate cancer (CRPC).
M2092 AZD3514 AZD3514 is a potent, small-molecule androgen receptor downregulator with potential anticancer cancer activity.
M1986 Andarine Andarine (GTx-007, S-4) is an orally active partial agonist for androgen receptors.
M1973 Ostarine (GTx-024) Ostarine (GTx-024 and MK-2866) is an investigational selective androgen receptor modulator (SARM) with Ki of 3.8 nM.
M1960 Bicalutamide Bicalutamide is an orally active non-steroidal androgen receptor antagonist (IC50 = 190 nM).
M1839 MDV3100 MDV3100 is an orally bioavailable, organic, non-steroidal small molecule targeting the androgen receptor (AR) with potential antineoplastic activity.
M1586 Norelgestromin Norgestimate and its metabolite norelgestromin possess weak androgen-like properties.

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