Inhibitors
Cat.No. | Name | Information |
---|---|---|
M1973 | Ostarine (GTx-024) | Ostarine (GTx-024 and MK-2866) is an investigational selective androgen receptor modulator (SARM) with Ki of 3.8 nM. |
M6033 | Dihydrotestosterone | Dihydrotestosterone is an androgen (male hormone). Specifically it's the strongest of the androgens. |
M6105 | Testosterone | Testosterone is an androgen, which binds the androgen receptor. |
M11350 | Triptophenolide | Triptophenolide is a colorless crystal isolated from the ethyl acetate extract of Triptophenolide. |
M10965 | ORM-15341 | ORM-15341 is a potent androgen receptor (AR) antagonist that acts on AR-HEK293 cells with an IC50 value of 38 nM. |
M10960 | Ralaniten | Ralaniten (EPI-002) is an effective and orally active androgen receptor N-terminal domain (AR-NTD) antagonist. Ralaniten inhibits AR transcriptional activity,IC50 The value is 7.4 μM. Ralanites can be used in the study of castration-resistant prostate cancer (CRPC). |
M10958 | JNJ-63576253 | JNJ-63576253 (TRC-253) is a potent and orally active complete antagonist of the androgen receptor against F877L mutant AR and wild-type AR in LNCaP cells IC50 The values are 37 and 54 nM, respectively. JNJ-63576253 can be used in the study of castration-resistant prostate cancer (CRPC). |
M10306 | Bavdegalutamide (ARV-110) | Bavdegalutamide (ARV-110) is an oral, specific androgen receptor (AR) PROTAC degrader. |
M9956 | Darolutamide | Darolutamide (ODM-201) is a new-generation, potent and selective androgen receptor (AR) inhibitor. |
M9149 | MI-136 | MI-136 inhibits DHT-induced expression of androgen receptor (AR) target genes. |
M9061 | Dehydroepiandrosterone | Dehydroepiandrosterone is an effective antiapoptotic factor. |
M8908 | ASC-J9 | ASC-J9, also known as GO-Y025 and Dimethylcurcumin, suppressesing castration-resistant prostate cancer growth through degradation of full-length and splice variant androgen receptors. |
M8128 | R1881 | R1881 (Metribolone) is an orally active, non-aromatisable androgen and anabolic steroid. |
M7561 | GSK-2881078 | GSK 2881078 is an androgen receptor regulator for the study of mental impotency. |
M6269 | Indacaterol | Indacaterol(Onbrez; Arcapta) is an ultra-long-acting β-adrenoceptor agonist. |
M6123 | Nandrolone phenylpropionate | Nandrolone phenylpropionate (NPP) is an anabolic-androgenic steroid. The low androgenicity and enhanced anabolic activity of NPP has shown to positively influence calcium metabolism and to increase bone mass in osteoporosis. |
M6122 | ChlordehydroMethyl Testosterone | A male hormone. |
M6121 | Testosterone phenylpropionate | Testosterone phenylpropionate is a synthetic anabolic-androgenic steroid (AAS) and an androgen ester. |
M6120 | Testosterone isocaproate | Testosterone isocaproate is an androgen. |
M6119 | Testosterone Enanthate | Androcur-treatment abolished testosterone-reduced cAMP, coupled with a changed expressional milieu of cAMP signaling elements. Results from in vitro experiments suggest that some of these effects are testosterone-AR dependent, while others could be due to disturbed LH and/or other signals. |
M6117 | Testosterone decanoate | Testosterone decanoate is an androgen. |
M6116 | Drostanolone Enanthate | Drostanolone is one of the most frequently detected anabolic androgenic steroids in doping control analysis. |
M6114 | Metandienone | Metandienone is a synthetic anabolic steroid that is prohibited in sports by the World Anti-Doping Agency (WADA). |
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