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Inhibitors
| Cat.No. | Name | Information |
|---|---|---|
| M1973 | Ostarine (GTx-024) | Ostarine (GTx-024 and MK-2866) is an investigational selective androgen receptor modulator (SARM) with Ki of 3.8 nM. |
| M6033 | Dihydrotestosterone | Dihydrotestosterone is an androgen (male hormone). Specifically it's the strongest of the androgens. |
| M6105 | Testosterone | Testosterone is an androgen, which binds the androgen receptor. |
| M5565 | Dexmedetomidine HCl | Dexmedetomidine Hydrochloride is an agonist of adrenergic alpha-2 receptor, which is used in veterinary medicine for its analgesic and sedative properties. |
| M20966 | Ligandrol (LGD-4033, VK-5211) | Ligandrol (LGD-4033, VK-5211) is a novel nonsteroidal, oral selective androgen receptor modulator with high affinity (Ki of ∼1 nM) and selectivity. |
| M20065 | WAY-298516 | WAY-298516 is a modulating rad51 |
| M14623 | UT-155 | UT-155 is a selective and potent androgen receptor (AR) antagonist, with a Ki of 267 nM for UT-155 binding to AR-LBD. |
| M14622 | Stanolone benzoate | Stanolone benzoate (Androstanolone benzoate) is a synthetic androgen and anabolic steroid. |
| M14621 | S-23 | S-23 is an orally active selective androgen receptor modulator (SARM) with a Ki of 1.7 nM. |
| M14620 | Vosilasarm | Vosilasarm (RAD140) is a potent, orally active, nonsteroidal selective androgen receptor modulator (SARM) with a Ki of 7 nM. Vosilasarm shows good selectivity over other steroid hormone nuclear receptors. |
| M14619 | MK-0773 | MK-0773 is a selective androgen receptor modulators (SARMs) that binds to AR with an IC50 of 6.6 nM. |
| M14618 | LY2452473 | LY2452473 is an orally bioavailable, selective androgen receptor modulator (SARM). |
| M14617 | GLPG0492 | GLPG0492 is a non-steroidal selective androgen receptor modulator (potency 12 nM). GLPG0492 has the potential for the research of musculo-skeletal diseases such as sarcopenia and cachexia. |
| M14616 | Dehydroisoandrosterone 3-acetate | Dehydroepiandrosterone 3-acetate is a testosterone/estrogen precursor and known modulator of vertebrate aggression. |
| M14615 | BMS-564929 | BMS-564929 is an androgen receptor (AR) agonist, binds to androgen receptor (AR) with a Ki of 2.11±0.16 nM. |
| M14614 | ACP-105 | ACP-105 is an orally available, selective amd potent androgen receptor modulator (SARM), with pEC50s of 9.0 and 9.3 for AR wild type and T877A mutant, respectively. |
| M14613 | 3,3'-Diindolylmethane | 3,3'-Diindolylmethane is a strong, pure androgen receptor (AR) antagonist. |
| M11350 | Triptophenolide | Triptophenolide is a colorless crystal isolated from the ethyl acetate extract of Triptophenolide. |
| M10965 | ORM-15341 | ORM-15341 is a potent androgen receptor (AR) antagonist that acts on AR-HEK293 cells with an IC50 value of 38 nM. |
| M10960 | Ralaniten | Ralaniten (EPI-002) is an effective and orally active androgen receptor N-terminal domain (AR-NTD) antagonist. Ralaniten inhibits AR transcriptional activity,IC50 The value is 7.4 μM. Ralanites can be used in the study of castration-resistant prostate cancer (CRPC). |
| M10958 | JNJ-63576253 | JNJ-63576253 (TRC-253) is a potent and orally active complete antagonist of the androgen receptor against F877L mutant AR and wild-type AR in LNCaP cells IC50 The values are 37 and 54 nM, respectively. JNJ-63576253 can be used in the study of castration-resistant prostate cancer (CRPC). |
| M10306 | Bavdegalutamide (ARV-110) | Bavdegalutamide (ARV-110) is an oral, specific androgen receptor (AR) PROTAC degrader. |
| M9956 | Darolutamide | Darolutamide (ODM-201) is a new-generation, potent and selective androgen receptor (AR) inhibitor. |
| M9149 | MI-136 | MI-136 inhibits DHT-induced expression of androgen receptor (AR) target genes. |
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