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 About 18 results found for searched term "CGRP Receptor" (0.128 seconds)

Cat.No.  Name Target
M2133 MK-3207 hydrochloride CGRP Receptor
MK-3207 hydrochloride is a potent CGRP receptor antagonist with IC50 of 0.12 nM.
M3618 MK-0974 CGRP Receptor
Telcagepant
MK-0974 (Telcagepant) is a highly potent, selective and orally bioavailable CGRP receptor antagonist with Ki values of 0.77 nM and 1.2 nM for human and rhesus CGRP receptors respectively.
M6504 Olcegepant (BIBN-4096) CGRP Receptor
BIBN-4096; BIBN 4096BS
Olcegepant (BIBN-4096) is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide (CGRP) receptor with IC50 of 0.03 nM and Ki of 14.4 pM for human CGRP.
M8322 SB-268262 CGRP Receptor
SB-268262 is a selective non-peptide antagonist at the CGRP1 receptor.
M10372 Vazegepant hydrochloride CGRP Receptor
Zavegepant, BHV-3500 hydrochloride
Vazegepant (BHV-3500) hydrochloride is a first-in-class, high affinity CGRP receptor antagonist (hCGRP Ki= 0.023 nM). Vazegepant hydrochloride may be useful in the effective treatment of lung inflammation associated with COVID-19.
M13931 Calcitonin Gene Related Peptide (CGRP) (83-119), rat TFA CGRP Receptor
Calcitonin Gene Related Peptide (CGRP) (83-119), rat (TFA) is a 37 amino acid calcitonin family of neuropeptide, acts through calcitonin receptor-like receptor (CRLR).
M13932 HCGRP-(8-37) CGRP Receptor
Human α-CGRP (8-37)
HCGRP-(8-37) is a human calcitonin gene-related peptide (hCGRP) fragment and also an antagonist of CGRP receptor.
M13933 MK-3207 CGRP Receptor
MK-3207 is a potent and orally bioavailable CGRP receptor antagonist (IC50= 0.12 nM; Ki= 0.024 nM); highly selective versus human AM1, AM2, CTR, and AMY3.
M13934 Olcegepant hydrochloride CGRP Receptor
BIBN-4096 hydrochloride; BIBN4096BS hydrochloride
Olcegepant hydrochloride (BIBN-4096 hydrochloride) is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and with a Ki of 14.4 pM for human CGRP.
M13935 Rat CGRP-(8-37) CGRP Receptor
Rat CGRP-(8-37) (VTHRLAGLLSRSGGVVKDNFVPTNVGSEAF) is a highly selective CGRP receptor antagonist.
M24721 Erenumab CGRP Receptor
Erenumab is a fully human monoclonal antibody. Erenumab inhibits the calcitonin gene–related peptide (CGRP) receptor. Erenumab can be used for the prevention of episodic migraine.
M24771 Eptinezumab CGRP Receptor
Eptinezumab is a human monoclonal antibody. Eptinezumab binds to calcitonin gene-related peptide (CGRP) and blocks its binding to the receptor. Eptinezumab can be used for the prevention of migraine in adults.
M28198 Vazegepant CGRP Receptor
Zavegepant; BHV-3500
Vazegepant (Zavegepant) is a first-in-class CGRP receptor antagonist with potential for acute studies in migraine.
M50213 CGRP antagonist 1 CGRP Receptor
CGRP antagonist 1 is a potent CGRP receptor antagonist with Ki and IC50 values of 1.7 nM and 5.7 nM, respectively.
M50214 AC 187 TFA Amyloid
AC 187 TFA is a potent, orally active and neuroprotective amylin receptor antagonist with an IC50 of 0.48 nM and a Ki of 0.275 nM. AC 187 TFA is more selective for amylin receptors than calcitonin and CGRP receptors.
M53227 [Tyr22] Calcitonin Gene Related Peptide, (22-37), rat CGRP Receptor
[Tyr22] Calcitonin Gene Related Peptide, (22-37), rat is a fragments 22-37 of rat calcitonin gene related peptide (CGRP), targeting CGRP receptor and adenylate cyclase.
M53230 Calcitonin Gene Related Peptide (CGRP) II, rat CGRP Receptor
Calcitonin Gene Related Peptide (CGRP) II, rat, a CGRP receptor activator, is a potent and long-lasting vasodilator.
M53900 Adrenomedullin (AM) (22-52), human CGRP Receptor
Adrenomedullin (AM) (22-52), human is an adrenomedullin receptor antagonist, and also antagonizes the calcitonin generelated peptide (CGRP) receptor in the hindlimb vascular bed of the cat.



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