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VU0410425 

Cat. No. M28203

All AbMole products are for research use only, cannot be used for human consumption.

VU0410425  Structure

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Quality Control & Documentation
Biological Activity

VU0410425 is an mGlu1 negative allosteric modulator. VU0410425 exhibits potent inhibitory activity for rat mGlu1 with an IC50 value of 140 nM. VU0410425 can be used for the research of central nervous system disorders.

Chemical Information
Molecular Weight 369.8
Formula C19H16ClN3O3
CAS Number 1341167-72-3
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Hyekyung P Cho, et al. ACS Chem Neurosci. A novel class of succinimide-derived negative allosteric modulators of metabotropic glutamate receptor subtype 1 provides insight into a disconnect in activity between the rat and human receptors

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  Catalog
Abmole Inhibitor Catalog




Keywords: VU0410425  supplier, GluR, inhibitors, activators

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