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Sutezolid

Cat. No. M8037

All AbMole products are for research use only, cannot be used for human consumption.

Sutezolid Structure
Synonym:

PNU-100480; U-100480; PF-02341272

Size Price Availability Quantity
5mg USD 70  USD70 In stock
10mg USD 120  USD120 In stock
25mg USD 240  USD240 In stock
50mg USD 380  USD380 In stock
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Quality Control & Documentation
Biological Activity

Sutezolid (PNU 100480) is an oxazolidinone antimicrobial. Sutezolid inhibits protein synthesis by inhibiting bacterial mRNA translation.

Sutezolid (PNU-100480) is a thiomorpholinyl analog of linezolid with superior efficacy against M. tuberculosis in the hollow-fiber, mouse, and whole-blood models.

Chemical Information
Molecular Weight 353.41
Formula C16H20FN3O3S
CAS Number 168828-58-8
Solubility (25°C) DMSO: 20 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Xia Yu, et al. In vitro Antimicrobial Activity Comparison of Linezolid, Tedizolid, Sutezolid and Delpazolid Against Slowly Growing Mycobacteria Isolated in Beijing, China

[2] Sarah Kim, et al. Pharmacokinetics of tedizolid, sutezolid, and sutezolid-M1 in non-human primates

[3] Aparna Bahuguna, et al. An overview of new antitubercular drugs, drug candidates, and their targets

[4] Christy Wyskiel. To be or not to be exclusive: the sutezolid story

[5] Jane Andrews. To be or not to be exclusive: the sutezolid story

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Keywords: Sutezolid, PNU-100480; U-100480; PF-02341272 supplier, Antibiotic, inhibitors, activators

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