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Sitagliptin

Cat. No. M5965

All AbMole products are for research use only, cannot be used for human consumption.

Sitagliptin Structure
Synonym:

MK0431

Size Price Availability Quantity
Free Sample (1-2 mg)  USD 0 In stock
50mg USD 40  USD40 In stock
100mg USD 55  USD55 In stock
200mg USD 70  USD70 In stock
Free Delivery on orders over USD 500 Bulk Inquiry?

Quality Control & Documentation
Biological Activity

Sitagliptin(MK 0431) is a potent inhibitor of DPP4 with IC50 of 19 nM in Caco-2 cell extracts.

Product Citations
Chemical Information
Molecular Weight 407.31
Formula C16H15F6N5O
CAS Number 486460-32-6
Solubility (25°C) DMSO 50 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Hartley P, et al. Drugs Aging. Efficacy and Tolerability of Sitagliptin Compared with Glimepiride in Elderly Patients with Type 2 Diabetes Mellitus and Inadequate Glycemic Control: A Randomized, Double-Blind, Non-Inferiority Trial.

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Keywords: Sitagliptin, MK0431 supplier, Dipeptidyl Peptidase, inhibitors, activators

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