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Trelagliptin

Cat. No. M2341

All AbMole products are for research use only, cannot be used for human consumption.

Trelagliptin Structure
Synonym:

SYR-472

Size Price Availability Quantity
10mM*1mL in DMSO USD 55  USD55 In stock
5mg USD 50  USD50 In stock
10mg USD 80  USD80 In stock
50mg USD 120  USD120 In stock
100mg USD 160  USD160 In stock
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Quality Control & Documentation
Biological Activity

Trelagliptin (SYR-472) is a highly selective once-weekly oral dipeptidyl peptidase-4 (DPP-4) inhibitor for type 2 diabetes. Trelagliptin (SYR-472) treatment produced clinically and statistically significant improvements in glycaemic control in patients with type 2 diabetes.

Product Citations
Chemical Information
Molecular Weight 357.38
Formula C18H20FN5O2
CAS Number 865759-25-7
Solubility (25°C) DMSO 60 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Inagaki N, et al. Lancet Diabetes Endocrinol. SYR-472, a novel once-weekly dipeptidyl peptidase-4 (DPP-4) inhibitor, in type 2 diabetes mellitus: a phase 2, randomised, double-blind, placebo-controlled trial.

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Keywords: Trelagliptin, SYR-472 supplier, Dipeptidyl Peptidase, inhibitors, activators

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