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SI-2 hydrochloride is a highly promising SRC-3 inhibitor (PPI) with acceptable oral availability, with IC50 values of 3-20 nM for breast cancer cell death.
| Molecular Weight | 301.77 |
| Formula | C15H16ClN5 |
| CAS Number | 1992052-49-9 |
| Solubility (25°C) | DMSO 3 mg/mL |
| Storage | 4°C, dry, sealed |
| Related Src-bcr-Abl Products |
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| KB SRC 4
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| Asciminib hydrochloride
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