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KX2-361 (KX-02) is a Src-kinase and tubulin polymerization inhibitor. KX2-361 shows anti-tumor activity and induces apoptosis of Glioblastoma (GBM) cell. KX2-361 shows good oral bioavailability and readily crosses the BBB in mice.
| Molecular Weight | 405.46 |
| Formula | C24H24FN3O2 |
| CAS Number | 897016-26-1 |
| Form | Solid |
| Solubility (25°C) | DMSO 9 mg/mL |
| Storage | 4°C, protect from light |
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