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S1P1 Agonist III is a potent and orally active S1P1 agonist with EC50 of 18 nM; no activity on S1P3.
Molecular Weight | 415.37 |
Formula | C21H16F3N3O3 |
CAS Number | 1324003-64-6 |
Form | Solid |
Solubility (25°C) | DMSO 62.5 mg/mL (ultrasonic) |
Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[1] Anthony Markham. Drugs. Ponesimod: First Approval
[2] Christopher Ma, et al. Drugs. Innovations in Oral Therapies for Inflammatory Bowel Disease
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