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Muraglitazar is a PPAR α/γ dual agonist for the research of type 2 diabetes and associated dyslipidemia. Muraglitazar shows potent activity in vitro at human PPARα (EC50 = 320 nM) and PPARγ(EC50 = 110 nM).
| Molecular Weight | 516.54 |
| Formula | C29H28N2O7 |
| CAS Number | 331741-94-7 |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
[2] Philip R Liebson. Prev Cardiol. Muraglitazar and the FDA: what constitutes drug safety?
[4] James M Brophy. JAMA. Selling safety--lessons from muraglitazar
[5] Daniela Barlocco. Curr Opin Investig Drugs. Muraglitazar (Bristol-Myers Squibb/Merck)
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