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ML381 (VU0488130) is a highly selective, central nervous system penetrant mAChR M5 orthogonal antagonist (IC50 = 450 nM; Ki = 340 nM). ML381 is unstable in rat plasma and can be mainly used as a molecular probe for in vitro and electrophysiological studies.
| Molecular Weight | 379.41 |
| Formula | C21H21N3O4 |
| CAS Number | 1623481-80-0 |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
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