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KZR-504 is a highly selective inhibitor of immunoproteasome low molecular mass polypeptide 2 (LMP2), with IC50s of 51 nM, 4.274 μM for LMP2 and LMP7, respectively. KZR-504 is of interest for the treatment of autoimmune disease.
| Molecular Weight | 413.42 |
| Formula | C21H23N3O6 |
| CAS Number | 1629052-78-3 |
| Form | Solid |
| Solubility (25°C) | DMSO 170 mg/mL (ultrasonic) |
| Storage | -20°C, protect from light, sealed |
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