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IOWH032 is a synthetic CFTR inhibitor with IC50 of 1.01 μM in CHO-CFTR cell based assays.
| Molecular Weight | 545.18 |
| Formula | C22H15Br2N3O4 |
| CAS Number | 1191252-49-9 |
| Solubility (25°C) | DMSO 90 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[2] Guiying Cui, et al. Potentiators exert distinct effects on human, murine, and Xenopus CFTR
[3] Eugenio L de Hostos, et al. Developing novel antisecretory drugs to treat infectious diarrhea
| Related CFTR Products |
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| GLPG2737
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