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TP-024 (FTBMT) is a selective GPR52 agonist with an EC50 of 75 nM. FTBMT (TP-024) (0.1-10 μM) increases intracellular cAMP levels in CHO cells expressing human, mouse, or rat GPR52, with pEC50s of 7.03, 6.85, and 6.87, respectively.
TP-024 (FTBMT) (3 or 10 mg/kg, 48 hours) improves recognition and spatial working memory in rats. FTBMT (TP-024) (3, 10, 30 mg/kg, 2 hours) stimulates neuronal activity in brain regions related to cognition.
| Molecular Weight | 392.35 |
| Formula | C19H16F4N4O |
| CAS Number | 1358575-02-6 |
| Solubility (25°C) | DMSO ≥ 40 mg/mL |
| Storage | 4°C, protect from light |
| Related GPR/FFAR Products |
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| CID1172084
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| ML 145
ML 145 is a selective and competitive human GPR35/CXCR8 antagonist with an IC50/EC50 of 20.1 nM. |
| PSN 375963 hydrochloride
PSN 375963 hydrochloride is a potent GPR119 agonist, with EC50s of 8.4 and 7.9 μM for human and mouse GPR119, respectively. |
All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.
Products are for research use only. Not for human use. We do not sell to patients.
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