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Edaglitazone

Cat. No. M29287

All AbMole products are for research use only, cannot be used for human consumption.

Edaglitazone Structure

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Quality Control & Documentation
Biological Activity

Edaglitazone is a potent, selective and orally active PPARγ agonist, with EC50s of 35.6 nM and 1053 nM for PPARα and PPARγ, respectively. Edaglitazone displays antiplatelet, antidiabetic and anti-hyperglycemic activity.

Chemical Information
Molecular Weight 464.56
Formula C24H20N2O4S2
CAS Number 213411-83-7
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Jinsai Shang, et al. Elife. Cooperative cobinding of synthetic and natural ligands to the nuclear receptor PPARγ

[2] Camila Muñoz-Gutiérrez, et al. Life Sci. Study of the interactions between Edaglitazone and Ciglitazone with PPARγ and their antiplatelet profile

[3] C Fürnsinn, et al. Br J Pharmacol. Chronic and acute effects of thiazolidinediones BM13.1258 and BM15.2054 on rat skeletal muscle glucose metabolism

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  Catalog
Abmole Inhibitor Catalog




Keywords: Edaglitazone supplier, PPAR, inhibitors, activators

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