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DS-6930 

Cat. No. M28026

All AbMole products are for research use only, cannot be used for human consumption.

DS-6930  Structure

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Quality Control & Documentation
Biological Activity

DS-6930 is a potent and selective agonist of PPARγ, with an EC50 of 41 nM. DS-6930 could robust reduce plasma glucose (PG), and with fewer PPARγ-related adverse effects than Rosiglitazone. DS-6930 can be used for the research of diabetes.

Chemical Information
Molecular Weight 403.43
Formula C23H21N3O4
CAS Number 1242328-82-0
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Tsuyoshi Shinozuka, et al. ACS Med Chem Lett. Structure-Activity Relationship Studies of 3- or 4-Pyridine Derivatives of DS-6930

[2] Tsuyoshi Shinozuka, et al. Bioorg Med Chem. Discovery of DS-6930, a potent selective PPARγ modulator. Part I: Lead identification

[3] Tsuyoshi Shinozuka, et al. Bioorg Med Chem. Discovery of DS-6930, a potent selective PPARγ modulator. Part II: Lead optimization

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  Catalog
Abmole Inhibitor Catalog




Keywords: DS-6930  supplier, PPAR, inhibitors, activators

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