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Domatinostat tosylate (4SC-202) is a selective class I HDAC inhibitor with IC50 of 1.20 μM, 1.12 μM, and 0.57 μM for HDAC1, HDAC2, and HDAC3, respectively. It also displays inhibitory activity against Lysine specific demethylase 1 (LSD1).
| Molecular Weight | 619.71 |
| CAS Number | 1186222-89-8 |
| Solubility (25°C) | DMSO ≥ 51 mg/mL |
| Storage | 2-8°C, dry, sealed |
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