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Bocidelpar

Cat. No. M29209

All AbMole products are for research use only, cannot be used for human consumption.

Bocidelpar Structure
Synonym:

ASP0367; MA-0211

Price and Availability

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Quality Control & Documentation
Biological Activity

Bocidelpar is a modulator of peroxisome proliferator-activated receptor delta (PPAR-δ). Bocidelpar improves mitochondrial biogenesis and function in Duchenne Muscular Dystrophy (DMD) muscle cells.

Chemical Information
Molecular Weight 460.49
Formula C25H27F3N2O3
CAS Number 2095128-20-2
Form Solid
Solubility (25°C) DMSO 150 mg/mL (ultrasonic)
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Mototsugu Ito, et al. Muscle Nerve. Single- and multiple-dose safety, tolerability, pharmacokinetic, and pharmacodynamic profiles of ASP0367, or bocidelpar sulfate, a novel modulator of peroxisome proliferator-activated receptor delta in healthy adults: Results from a phase 1 study

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Keywords: Bocidelpar, ASP0367; MA-0211 supplier, PPAR, inhibitors, activators

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