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Bikinin

Cat. No. M8228

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Bikinin Structure
Synonym:

Abrasin

Size Price Availability Quantity
10mM*1mL in DMSO USD 28  USD28 In stock
5mg USD 25  USD25 In stock
10mg USD 40  USD40 In stock
50mg USD 125  USD125 In stock
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Quality Control & Documentation
Biological Activity

Bikinin is a strong activator of brassinosteroid (BR) signaling. It is an Arabidopsis GSK-3 Inhibitor, an Arabidopsis SHAGGY-related Kinase Inhibitor, and a GSK-3-like Kinase BIN2 Inhibitor. Bikinin directly inhibits BIN2 (group II GSK3s) by interfering with ATP binding. Bikinin is specific toward a subset of Arabidopsis GSK3 kinases including BIN2 and ASK α, γ, ε, ι, and θ.

Chemical Information
Molecular Weight 273.08
Formula C9H9BrN2O3
CAS Number 188011-69-0
Solubility (25°C) DMSO ≥ 30 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Wilfried Rozhon, et al. Inhibitors of Brassinosteroid Biosynthesis and Signal Transduction

[2] Takema Sasaki, et al. Imaging of Developing Metaxylem Vessel Elements in Cultured Hypocotyls

[3] Hye Jo Min, et al. OsBZR1 turnover mediated by OsSK22-regulated U-box E3 ligase OsPUB24 in rice BR response

[4] Kyoko Yamazaki, et al. Suppression of DELLA signaling induces procambial cell formation in culture

[5] Wilfried Rozhon, et al. Bikinin-like inhibitors targeting GSK3/Shaggy-like kinases: characterisation of novel compounds and elucidation of their catabolism in planta

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  Catalog
Abmole Inhibitor Catalog




Keywords: Bikinin, Abrasin supplier, GSK-3, inhibitors, activators

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