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ACT-660602

Cat. No. M21323

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ACT-660602  Structure
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Biological Activity

ACT-660602 is an oral chemokine receptor CXCR3 antagonist with an IC50 of 204 nM. It is being developed for use in autoimmune diseases.

Chemical Information
Molecular Weight 534.48
Formula C20H20F6N8OS
CAS Number 1646267-59-5
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Emmanuel A Meyer, et al. J Med Chem. Discovery and In Vivo Evaluation of ACT-660602: A Potent and Selective Antagonist of the Chemokine Receptor CXCR3 for Autoimmune Diseases

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Keywords: ACT-660602 supplier, CXCR, inhibitors, activators

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