Activator
| Cat.No. | Name | Information |
|---|---|---|
| M45066 | Ulotaront HCl | Ulotaront HCl is a first-in-class, orally active, CNS-active TAAR1 agonist for studies related to schizophrenia. |
| M29285 | Ralmitaront | Ralmitaront (RO6889450), a potent and orally active partial agonist of the trace amine-associated receptor 1 (TAAR1), acts as a neuroleptic agent. Ralmitaront can be used for the research of neuro-related diseases, such as schizophrenia (SCZ), schizoaffective disorder, and negative symptoms. |
| M20404 | Tryptamine | Tryptamine is a monoamine alkaloid and may play a role as a neuromodulator or neurotransmitter. It is an agonist of hTAAR1. It acts as a non-selective serotonin receptor agonist and serotonin-norepinephrine-dopamine releasing agent (SNDRA). |
| M28237 | RO5263397 | RO5263397 is a potent, selective, and orally available TAAR1 agonist, with EC50s of 17 and 35 nM for human TAAR1 and rat TAAR1, respectively. RO5263397 regulates wakefulness and EEG spectral composition. Antidepressant-like effect. |
| M27714 | RO5166017 | RO5166017 is an orally active and species-crosses TAAR1 agonist, with Ki values of 1.9 nM, 2.7 nM, 31 nM and 24 nM for mouse, rat, human and cynomolgus monkey, respectively. |
| M27700 | RO5203648 | RO5203648 is a potent and highly selective partial agonist of TAAR1 (Trace amine-associated receptor 1) with high affinity. RO5203648 demonstrates a novel paradigm for neuropsychiatric research. |
| M21226 | Ulotaront | Ulotaront (SEP-856) is a first-in-class, orally active, CNS-active TAAR1 agonist for use in studies related to schizophrenia. |
| M8721 | RO5256390 | RO5256390 is a selective agonist of trace amine-associated receptor 1 (TAAR1) and a negative modulator of dopamine transmission for studies related to schizophrenia and bulimia. |
| M8504 | EPPTB | EPPTB is a potent, selective trace amine-associated receptor 1 (TAAR1) antagonist with an IC50 value of 28 nM for mouse TAAR1. EPPTB is less selective in rats and humans, with IC50 values of 4539 nM and 7487 nM, respectively. |
| M8327 | D,L-Metanephrine hydrochloride | Metanephrine is an endogenous metabolite of epinephrine, formed by catechol-O-methyltransferase activity, as well as a biomarker of cancer and can be used to diagnose pheochromocytoma. In addition, Metanephrine is a potent agonist of the trace amine-associated receptor TAAR1. |
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