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EPPTB is a potent, selective trace amine-associated receptor 1 (TAAR1) antagonist with an IC50 value of 28 nM for mouse TAAR1. EPPTB is less selective in rats and humans, with IC50 values of 4539 nM and 7487 nM, respectively.
| Molecular Weight | 378.39 |
| Formula | C20H21F3N2O2 |
| CAS Number | 1110781-88-8 |
| Solubility (25°C) | DMSO 20 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
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