Inhibitor
| Cat.No. | Name | Information |
|---|---|---|
| M3510 | Mifepristone | Mifepristone is a remarkably active antagonist of progesterone receptor and glucocorticoid receptor with IC50 of 0.2 nM and 2.6 nM, respectively. |
| M30085 | Allylestrenol | Allylestrenol is an anabolic steroid with progesterone activity and potential physiologic function as a progesterone receptor agonist that can be used in studies related to preterm labor. |
| M14796 | Medroxyprogesterone | Medroxyprogesterone is a progestin, a synthetic variant of the human hormone progesterone and a potent progesterone receptor agonist. |
| M8390 | Nestorone | Nestorone is a potent progesterone receptor agonist with no androgenic, estrogenic, or glucocorticoid-like activities. |
| M6043 | Ulipristal acetate | Ulipristal acetate(CDB2914) is a novel selective progesterone receptor modulator (SPRM) for the treatment of benign gynecological conditions such as uterine myoma. |
| M5357 | 17-Hydroxyprogesterone | 17-Hydroxyprogesterone (17-OHP) is an endogenous progestogen as well as chemical intermediate in the biosynthesis of other steroid hormones, including the corticosteroids and the androgens and the estrogens. |
| M3346 | Levonorgestrel | Levonorgestrel is a synthetic progestogen used as an active ingredient in some hormonal contraceptives. |
| M3100 | Ulipristal | Ulipristal is a selective SPRM for emergency contraception after an unprotected intercourse or contraceptive failure. |
| M2887 | Norethindrone | Norethindrone is a synthetic progestin, which mimic the actions of the endogenous ovarian hormone progesterone. |
| M2692 | Ethynodiol diacetate | Ethynodiol diacetate is one of the first synthetic progestogens used in contraceptive pills. |
| M2658 | Dydrogesterone | Dydrogesterone is an orally active progestogen which acts directly on the uterus, producing a complete secretory endometrium in an estrogen-primed uterus. |
| M2377 | Altrenogest | Altrenogest is a progestogen structurally related to veterinary steroid trenbolone. |
| M2260 | Gestodene | Gestodene is a synthetic progestin used as a contraceptive. |
| M2232 | Dienogest | Dienogest is an orally-active semisynthetic, steroidal progestogen (or progestin). |
| M43604 | Trimegestone | Trimegestone (RU 27987) is an orally active 19-norpregnane progestin. |
| M30327 | Nomegestrol | Nomegestrol is a potent and orally available progestin, acts as a selective full progesterone receptor agonist, with a Kd of 5.44 nM for rat uterine progesterone receptor, and has moderate antiandrogenic activity and strong antiestrogenic activity. |
| M30029 | Cridanimod | Cridanimod is a potent progesterone receptor (PR) activator mediated through induction of IFNα and IFNβ expression. Cridanimod is a small-molecule immunomodulator and interferon inducer. |
| M29084 | Asoprisnil | Asoprisnil (J867), a selective progesterone receptor modulator, exhibits mixed progesterone agonist and antagonist effects on various progesterone targeted tissues in animal and human. |
| M14797 | Tanaproget | Tanaproget (NSP-989) is a novel nonsteroidal progesterone receptor agonist which can bind to the PR from various species with a higher relative affinity than reference steroidal progestins. |
| M8119 | PF-02413873 | PF-02413873 is a potent, selective and fully competitive non-steroidal progesterone receptor (PR) antagonist that blocks progesterone binding and PR nuclear translocation. |
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