Progesterone Receptor Inhibitors | Kinase Inhibitors on Progesterone Receptor Signaling Pathways

Progesterone Receptor Progesterone receptor (PR)

Inhibitor

Cat.No.	Name	Information
M3510	Mifepristone	Mifepristone is a remarkably active antagonist of progesterone receptor and glucocorticoid receptor with IC50 of 0.2 nM and 2.6 nM, respectively.
M8119	PF-02413873	PF-02413873 is a potent, selective and fully competitive non-steroidal progesterone receptor (PR) antagonist that blocks progesterone binding and PR nuclear translocation.

Cat.No.

Name

Information

M3510

Mifepristone is a remarkably active antagonist of progesterone receptor and glucocorticoid receptor with IC50 of 0.2 nM and 2.6 nM, respectively.

M8119

PF-02413873

PF-02413873 is a potent, selective and fully competitive non-steroidal progesterone receptor (PR) antagonist that blocks progesterone binding and PR nuclear translocation.